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(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
N,1-dimethyl-6-oxo-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,6-dihydropyridazine-3-carboxamide
2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-[3-(2-{[cyclohexyl(methyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
N-methyl-5-(propan-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
1-cyclopropanecarbonyl-N-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
5,8-dichloro-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
3-{[2-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}phenol
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[5-(methoxymethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-chloro-4-fluoro-5-methylphenyl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(pyridin-3-ylmethyl)acetamide
5-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-fluoro-4-methylquinoline
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
5-methyl-2-[4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
(4aS,8aS)-4a-hydroxy-N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]-decahydroisoquinoline-2-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(pyridin-4-yl)piperidine-4-carboxylic acid
(1R,9aR)-1-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
14-(4-methyl-2-oxo-2H-chromen-7-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
(2S,4R)-4-amino-N-methyl-1-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}pyrrolidine-2-carboxamide
N-ethyl-5-(1H-indol-1-ylmethyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
6-[(E)-2-phenylethenyl]-1H-[1,2,3]triazolo[4,5-b]pyridine
8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-ethyl-N4-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
N-[(1-benzylpyrrolidin-3-yl)methyl]oxan-4-amine
[6-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridin-2-yl]methanol
4-[1-(4-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydropyridin-2-one
N-({5-[(5-cyclohexylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-ethyl-1H-indole
1-(2-methylpropyl)-N,5-bis(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[4-(2-methoxyphenoxy)piperidin-1-yl]-4-oxobutane-1-sulfonamide
1-[2-(1H-imidazol-1-yl)propyl]-4-(2-phenylphenyl)-1H-1,2,3-triazole
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
1-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
1-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(prop-2-en-1-yl)urea
ethyl (1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
3-methyl-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
(3R,5R)-N-[2-(1H-indol-3-yl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
1-({4-methyl-5-[1-(pyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-{3-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]phenyl}ethan-1-one
[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl](2-methoxyethyl)methylamine
2-[(3-methoxyphenyl)amino]-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]butanamide
3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroisoquinolin-1-one