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[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(2-phenylphenyl)methyl]pyrrolidin-3-yl]methanol
[(5-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}thiophen-3-yl)methyl]dimethylamine
4-ethyl-3-{[1-(naphthalen-1-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2E)-3-(2-chlorophenyl)-N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)prop-2-enamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4,5-trimethoxybenzamide
3-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidine-1-carboxamide
2-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
3-(2-methoxy-5-methylphenyl)-5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazole
1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]-4-(4-chlorophenyl)piperidin-4-ol
2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)-N-{[2-(trifluoromethyl)phenyl]methyl}pyridine-3-carboxamide
methyl 4-[5-methyl-4-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)-1,3-oxazol-2-yl]benzoate
1-(2-hydroxyethyl)-N-methyl-N-[2-(phenylsulfanyl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-{4-[2-(propan-2-yl)-1H-imidazol-1-yl]butyl}pyridine
N-methyl-2-(4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrimidin-4-amine
1-[2-(difluoromethoxy)benzoyl]-2-(4-fluorophenyl)pyrrolidine
7-[(3-methoxyphenyl)methyl]-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-4-(1H-1,2,4-triazol-3-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}benzamide
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3S,4R)-1-(5-methoxyfuran-2-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
(2S,4R)-4-[(adamantan-2-yl)amino]-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N5-cyclooctyl-N3-methyl-4-oxo-N3-(propan-2-yl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-1,4-diazepane-6-carboxylic acid
4-benzyl-3-ethyl-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-5-one
3-chloro-N-(2-methoxyethyl)-4-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
3-(oxolan-3-yl)-5-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1,2,4-oxadiazole
N-{1-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
N-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
6-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
(2R,6R)-11-methoxy-4-(3,3,4,4-tetrafluorobutyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
5-cyclopropanecarbonyl-1'-(5-fluoro-2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-({2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}methyl)benzonitrile
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(4-{[1-(quinolin-5-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-(3-methoxypropyl)-1-methyl-5-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(propylsulfanyl)ethan-1-one
1-[(5-fluoro-2-methoxyphenyl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-methyl-4-[5-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)thiophen-2-yl]but-3-yn-2-ol
N-(butan-2-yl)-1-(4,7-dimethylquinazolin-2-yl)azepan-4-amine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-3-yl)acetamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-(pyrrolidine-1-carbonyl)piperazine
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine-4-carboxylic acid
4-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrimidin-2-amine
4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,3,5-trimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-benzofuran-2-carboxamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
N-benzyl-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)acetamide