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4-fluoro-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
(1S,4S)-2-(2-fluorophenyl)-5-(3-phenylpropyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
5-(3-fluorophenoxymethyl)-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
3-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-N-(pyridin-3-yl)propanamide
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}piperidine
N-butyl-3-cyclopentaneamido-4-methyl-N-(pyridin-3-ylmethyl)benzamide
N-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
8-[(2-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-7-methyl-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
ethyl 3-(2-methoxyethyl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidine-3-carboxylate
1-ethyl-4-{[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-[2-methyl-5-(3-methylbutanamido)phenyl]-5-oxopyrrolidine-3-carboxylic acid
8-({3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[1-(pyridin-3-yl)pentyl]acetamide
1-[(4-fluorophenyl)methyl]-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1,3-thiazole
1-(3-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}piperidin-1-yl)-2-methoxyethan-1-one
1-{3-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenyl}ethan-1-one
3-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
1-(2,3-dihydro-1H-inden-4-yl)-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
1-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}piperidine-4-carboxamide
4-({1-[(5-phenylthiophen-2-yl)methyl]piperidin-2-yl}methyl)morpholine
N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]-3-(2-oxopyrrolidin-1-yl)propanamide
1-{1-[(2-fluoro-5-methoxyphenyl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-[2-(propan-2-yloxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2,3-dimethoxyphenyl)-4-(4-ethoxyphenyl)-1H-imidazole
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
6-benzyl 4a-ethyl (4aS,8aR)-decahydro-1,6-naphthyridine-4a,6-dicarboxylate
(3aR,5R,6S,7aS)-2-[2-(trifluoromethyl)benzoyl]-octahydro-1H-isoindole-5,6-diol
2-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]morpholin-3-yl}-N-(pyridin-3-yl)acetamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-(2-chloro-5-methylphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
N4-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methylphenyl)ethan-1-one
N,N-dimethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-{2-[2-(4-fluorophenyl)morpholin-4-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
methyl 3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)benzoate
(1S,9aR)-1-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
3-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}urea
N-(2-fluoro-4-methylphenyl)-2-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}acetamide
3-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}-4H-chromen-4-one
3-cyclopropyl-N-[2-(dimethylsulfamoyl)ethyl]-1H-pyrazole-5-carboxamide
2-cyclopropyl-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1,3-benzoxazole-6-carboxamide