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1'-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(methylsulfanyl)pyridine-3-carboxamide
4-[(2-chlorophenyl)methyl]-1-[3-(furan-2-yl)benzoyl]-1,4-diazepan-5-one
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
2-(carbamoylamino)-N-[(3R,4S)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-[2-(2-methylphenyl)ethyl]-1-(1H-pyrazole-4-carbonyl)piperidine
1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazole
N-ethyl-N-(2-hydroxyethyl)-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
(4aS,8aR)-6-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)pyrimidine
(3S,4R)-N,N-dimethyl-4-propyl-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]pyrrolidin-3-amine
6-(3-fluorophenyl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-(4-methylphenoxy)piperidin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-4-phenoxybutanamide
5-(1H-imidazol-2-yl)-4-phenyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-imidazole
2-[3-(1-methoxypropyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetic acid
4-(1,3-benzothiazol-2-yl)-2-[(2-ethylpiperidin-1-yl)methyl]phenol
4-benzyl-1-[(3-fluoro-4-methylphenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-4-yl}piperidin-4-ol
1-[7-(3-chlorophenyl)-9-(pyridin-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
2-(1-benzofuran-2-yl)-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid
2-(benzyloxy)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
N-(2,3-dihydro-1-benzofuran-3-yl)-2,5,6-trimethylpyrimidin-4-amine
3-(2-methyl-5-oxopyrrolidin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
1'-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
2-{4-methyl-2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]phenoxy}acetamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-3-yl]methanol
4-{5-[2-(3-fluorophenyl)ethyl]-1-methyl-1H-1,2,4-triazol-3-yl}pyridine
N-[2-(pyridin-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-4-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}benzamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(4H-1,2,4-triazol-4-yl)propanamide
(3R,5R)-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-3-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]urea
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
methyl 3-({[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate
5-(4-methoxy-2,3-dimethylphenyl)-3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
5-chloro-N-(1H-imidazol-2-ylmethyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
4,6-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
N-cyclopropyl-1-phenyl-N-(thiophen-3-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
2-{[4-amino-6-(4-methyl-1,4-diazepan-1-yl)pyrimidin-2-yl]sulfanyl}-N,N-dimethylacetamide
(4aS,7aR)-N-tert-butyl-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]propanamide
N-[1-(pyridin-2-yl)propan-2-yl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide