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methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2-{7-[(1-propyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-({5-[(2-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-1H-1,3-benzodiazole-5-carbonitrile
2-(5-methyl-1,2-oxazol-3-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
3-{[(1H-1,3-benzodiazol-2-ylmethyl)amino]methyl}-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
2-(2-{5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrrol-1-yl)pyrimidine
3-(benzenesulfonyl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-fluoro-6-methoxybenzoyl)-3-methylpiperidine
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
1-(4-chlorophenyl)-N-[(1,1-dioxo-1λ6-thian-4-yl)methyl]cyclobutane-1-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-methyl-1,3-thiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-ol
(1S,5R)-6-(6-methylpyridine-3-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-1-(1,4-dimethyl-1H-indole-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1,3-thiazole-4-carboxamide
5-benzyl-5-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
6-methyl-N-(morpholin-2-ylmethyl)-2-propylpyrimidin-4-amine
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(1S,6R)-3-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-ethyl-6-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-N-methylpyridine-3-carboxamide
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethyl-1H-pyrrole-2-carboxamide
methyl 8-[(4-fluoro-3-methoxyphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2-methoxyethyl)-2-(pyrrolidin-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-butyl-8-(1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(2-ethylpyrimidine-5-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-benzyl-9-[(2R)-2,5-diaminopentanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
N-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N2,N2,N4,N4-tetramethyl-7-(3-propyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-3-phenyl-1,2,4-oxadiazole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
6-(2-aminoethyl)-2-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
3-ethoxy-1-[4-(4-fluorophenoxy)piperidin-1-yl]propan-1-one
1-{1-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]piperidin-4-yl}pyrrolidin-2-one
1-[(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
4-methyl-5-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-(4-methoxybenzoyl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-3-yl]urea
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(cyclobutylmethyl)(oxolan-2-ylmethyl)amine
1-(3-fluorophenyl)-6,6-dimethyl-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-{5-[6-amino-5-cyano-4-(pyridin-4-yl)pyridin-2-yl]thiophen-3-yl}acetic acid
methyl (2S)-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidine-2-carboxylate
3,5-difluoro-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
3-[4-(3-methoxypropyl)piperazine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one