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N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
1,3-dimethyl-4-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-one
1-[(2-methoxyphenyl)methyl]-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
N-[(1-benzylpiperidin-4-yl)methyl]-3-ethyl-N-methyl-1H-pyrazole-4-carboxamide
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-[(3-fluoro-4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(carbamoylmethyl)-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
2-methoxy-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoline
(1S,6R)-9-{[2-(furan-2-yl)phenyl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
N-{1-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl 3-(4-{[(4aS,7aR)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
N-[(2R,3R)-1'-[(4-fluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
8-fluoro-3-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(3-carbamoylpyridin-2-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
3-[2-(4-methoxyphenyl)ethyl]-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidine
N2-[1-(9H-purin-6-yl)piperidin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-N-[(2,5-dimethoxyphenyl)methyl]acetamide
1-{1-[(2-chloro-3,6-difluorophenyl)methyl]azetidin-3-yl}-2-methylpiperidine
1-[(3-fluorophenyl)methyl]-N-methyl-6-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxamide
N-[(2S,4R,6S)-2-(3-cyanophenyl)-6-(2-methylpropyl)oxan-4-yl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N5-cycloheptyl-1-cyclopropyl-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-chlorophenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,5R)-6-{[4-(1H-imidazol-1-yl)phenyl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]-1-[(1S)-1-(3-methylpyridin-2-yl)ethyl]urea
(2S,4S)-4-amino-1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(methylsulfanyl)propanamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-4-phenyl-N-(pyridin-4-ylmethyl)benzamide
1-(1-benzofuran-5-ylmethyl)-4-(2-methoxybenzoyl)piperazine
(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
2,3,6-trimethyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]quinoline-4-carboxamide
methyl(pyrazin-2-ylmethyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
1-(3-phenylpiperazin-1-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
methyl 6-(but-3-enoyl)-2-{[(4-chlorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3-{2-[1-(3-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
7-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-2-yl}ethan-1-ol
6-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
3-(3-fluorophenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(pyridin-4-yl)quinoline
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-6-methoxypyrimidin-4-amine
5-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,2-oxazol-3-amine
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-5-propyl-1,2-oxazole-3-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-(4-methyl-1,4-diazepan-1-yl)acetamide
1,4-dimethyl 2-[(1-{4-[2-(3-chlorophenyl)acetamido]phenyl}piperidin-4-yl)amino]butanedioate