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methyl 6-[(2-fluoro-4-methoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-({1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)propane-1-sulfonamide
1-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
N-[(2R,3R)-1'-[(4-ethylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-(3-hydroxypropyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
3-(2-methoxyphenyl)-1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
{4-[(4-methoxyphenyl)methyl]-1-(quinolin-2-yl)piperidin-4-yl}methanol
2-(dimethylamino)-2-(4-fluorophenyl)-N-(3-methoxypropyl)acetamide
N-[(3S,4R)-1-[(5-methylthiophen-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(3aR,6aR)-2-methyl-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
N-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
benzyl N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}carbamate
2-[(3-chlorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
1-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]furan-2-carboxamide
1-ethyl-N,5-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
[(4-ethylphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(4-ethylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridin-3-amine
[(3R,4S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(3S,5R)-1-(2-methylpropyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(2S)-2-{[5-(carboxymethyl)pyrimidin-4-yl]amino}-3-(1H-indol-3-yl)propanoic acid
2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)acetamide
4'-(2,2-dimethylpropyl)-1-(furan-3-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{[4-(1-phenylethyl)-5-(pyrazin-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-ethyl-8-(5-phenyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-(4-methylphenoxymethyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
5-methyl-1-(4-methylphenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
3-(3-methoxyphenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(2-methylfuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-(2-methyl-1H-indol-3-yl)-N-[1-(pyridin-4-yl)ethyl]acetamide
2-methoxy-1-[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
1-ethyl-4-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}pyrrolidin-2-one
N-methyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxamide
N-(3-methoxypropyl)-1-methyl-5-[(3-methylquinoxalin-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-cyclopropyl-3-[2-(3,4-dimethylpiperazin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3S,4S)-3-hydroxy-4-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-1-yl]ethan-1-one
5-{2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[(3-methoxyphenyl)methyl]-4-(quinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
2-amino-4-(thiophen-2-yl)-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(2-methylpropyl)amine
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-4-(piperidin-1-yl)butanamide
8-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-[2-(5-cyclopropyl-1H-pyrazol-1-yl)ethyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine