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N-methyl-5-phenyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2,4-oxadiazol-3-amine
methyl 2-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}benzoate
(3R,4R)-1-(2,4-difluoro-3-methoxybenzoyl)-4-(hydroxymethyl)piperidin-3-ol
2-(1-benzofuran-2-yl)-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetic acid
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-ol
4-methyl-2-{[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}-1,2-dihydrophthalazin-1-one
4-benzyl-3-ethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,4-diazepan-5-one
2-[(4aR,7aS)-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
3-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1,2-oxazole
3-(1-{1-[1-(2-methoxyphenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
1-[4-({cyclopropyl[(2-methoxyphenyl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-(1,4-dioxan-2-ylmethyl)-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamide
methyl 4-oxo-4-(4-{4-[(2-phenylethyl)carbamoyl]phenoxy}piperidin-1-yl)butanoate
ethyl 4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazine-1-carboxylate
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-methoxypyridine-3-carboxamide
1-(carbamoylmethyl)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]quinoline-3-carboxamide
2-(pyridin-3-yl)-1-[4-(pyridin-3-yloxy)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
4-benzyl-1-[(3-fluorophenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetyl]-1,4-diazepan-5-one
2-(2-chloro-6-fluorobenzamido)-7-oxo-N-[1-(thiophen-2-yl)propyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
(5S,9aS,9bS)-5-(2,1,3-benzothiadiazol-5-yl)-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-(thiophene-2-carbonyl)piperidin-4-amine
3-{4-[(3-chloropyridin-4-yl)methyl]piperazin-1-yl}-1,2-benzothiazole
3-{1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-1,2,3-triazol-4-yl}phenol
3-(2-chlorophenyl)-N-cyclobutyl-3-(3-hydroxyphenyl)propanamide
N-[(2R,3R)-2-methoxy-1'-(quinolin-5-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
5-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]pyridine-2-carbonitrile
N-[2-(oxan-2-yl)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1'-(2-methyl-5-propylpyrimidin-4-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(1-benzofuran-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-(1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-ethyl-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]butan-1-one
1-[2-(propan-2-yl)pyrimidine-5-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]pyridine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(morpholine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(1,2-oxazol-5-ylmethyl)-2-(pyridin-4-yl)quinoline-4-carboxamide
2-cyclohexyl-5-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidine
4-[(2-fluorophenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-methoxy-3-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(4aR,8aR)-7-[3-(dimethylamino)benzoyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(4aS,7aR)-1-(3-chlorobenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
2,4-dimethoxy-6-(2-methoxy-5-methylphenyl)-1,3,5-triazine