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N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
1-[2-(benzyloxy)ethyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-cyclopropyl-3-ethoxy-N-[(3-ethoxyphenyl)methyl]propanamide
1-[(3-methoxyphenyl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-[4-(pyridin-4-yloxy)piperidin-1-yl]pyrimidine
1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-2,6-dione
(3R,4R)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
5-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}quinoxaline
1-[4-(2-fluorophenyl)benzoyl]-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-(3-cyclopentylpropanoyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-N-(4-fluorophenyl)piperidin-3-amine
2-(3-methoxyphenyl)-6-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,3-benzoxazole
2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-4-(propan-2-yl)-1,4-diazepane
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
5-({2-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
3-(4-benzyl-1H-pyrazol-5-yl)-1-(4-chloro-1H-pyrazole-3-carbonyl)piperidine
2-cyclobutyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(2-methoxyacetamido)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
2-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
2-(1-ethylpiperidin-4-yl)-1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}ethan-1-one
(2S,4R)-4-amino-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,4R)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-cyclobutyl-3-methylpiperidin-4-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carboxamide
[(2S)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
2-{4-[1-(4-chlorophenyl)cyclobutanecarbonyl]morpholin-3-yl}-N-methylacetamide
4-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}butan-2-ol
1-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-4-yl}pyrrolidin-2-one
N-[3-(4-methoxyphenyl)propyl]-6-(2-methyl-1,4-oxazepan-4-yl)pyridine-3-carboxamide
3-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrrolidin-3-ol
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]urea
3-(5-methyl-4H-1,2,4-triazol-3-yl)-N-(1,2,3,4-tetrahydroquinolin-1-yl)propanamide
(2S,4S)-4-amino-1-(2-cyclopropylquinoline-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
[3-(1H-imidazol-1-yl)propyl][(4-methyl-1H-imidazol-5-yl)methyl](pyridin-3-ylmethyl)amine
6-{3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
methyl[1-(pyrazin-2-yl)propan-2-yl]{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
5-methyl-4-[(oxolan-3-yl)amino]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
(2S)-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)pentan-1-one
4-{5-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
7,7-dimethyl-2-{1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,7aR)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(phenylamino)pyrimidine-5-carboxamide
1-(ethanesulfonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(2-methyl-1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
4-[3-(2-methylphenyl)benzoyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(1-{[methyl({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl})amino]methyl}cyclopropyl)methanol