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3-[(3-acetamidopyrrolidin-1-yl)methyl]-N-(3-methyl-1,2-thiazol-5-yl)benzamide
1-(2-fluorophenyl)-4-[4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]piperidin-4-ol
2,3,5-trimethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-methoxy-N-methyl-4-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4H-pyran-2-carboxamide
1-[4-(methylsulfanyl)phenyl]-3-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-4-amine
methyl 3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethoxy]benzoate
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[2-(azepan-1-yl)ethyl]-N,4-dimethylpyrimidin-2-amine
N-(1-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}propan-2-yl)acetamide
N-[(1-methylpiperidin-4-yl)methyl]-3-(prop-2-en-1-yloxy)benzamide
N-[2-methyl-6-(propan-2-yl)phenyl]-2-[(quinolin-3-ylmethyl)amino]acetamide
N-cyclopentyl-4-methyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1,2,5-oxadiazole-3-carboxamide
5-ethyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-2-amine
N,1,2-trimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-imidazole-4-sulfonamide
2-(4-chloro-2-methylphenoxy)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
3-cyclopropyl-N-[2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
1-(4-methylphenyl)-4-[4-(piperidin-1-yl)pentanoyl]piperazin-2-one
2-amino-7-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(1-methyl-1H-pyrazol-4-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}propan-1-one
3-{5-cycloheptyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopropylpropanamide
N-[(3-chlorophenyl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
(3S,4R)-3-ethyl-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-methylpiperidin-4-ol
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
7-cyclohexyl-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-({7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
4-(1,7-dimethyl-1H-indole-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
(1S,3R)-N1,1,2,N2,N3,3-hexamethyl-N1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]cyclopentane-1,3-dicarboxamide
1-[5-(dimethylcarbamoyl)pyridin-2-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(2,6-difluorophenyl)methyl]-N-[1-(4-fluorophenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-[1-(4-methoxyphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
3-(3,4-dimethylphenyl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(2,5-dimethylthiophen-3-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-methylthiophene-2-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-{[4-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
N-methyl-5-(oxolan-2-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}thiophene-2-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(phenylsulfanyl)acetamide
8-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]urea
2,2-dimethyl-4-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide