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4-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-4H-1,2,4-triazole
1-ethyl-4-{[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1H-pyrrole-2-carbonitrile
(3S,4R)-N,N-dimethyl-4-propyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-amine
1-[(2-aminopyridin-3-yl)methyl]-4-(isoquinolin-1-yl)-1,4-diazepan-6-ol
2-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)-1H-indole
N-[(2R,3R)-1'-(isoquinolin-5-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-{[(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N5-[(1R)-1-(4-methoxyphenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-methoxy-2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenol
4,4,4-trifluoro-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,2-oxazole-3-carboxamide
1-(furan-2-ylmethyl)-4-[3-(3-methoxypropyl)piperidine-1-carbonyl]piperidine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-[(1-cyclohexanecarbonylpyrrolidin-2-yl)formamido]-N-(1,3-thiazol-2-yl)acetamide
(4aS,7aR)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[5-(methoxymethyl)furan-2-carbonyl]-4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
3-{1-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]piperidin-4-yl}phenol
ethyl 4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
1-methyl-4-phenyl-3-{1-[2-(pyridin-4-yl)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2,6-difluoro-4-methoxyphenyl)methyl]-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-4-amine
1-{6-[4-(1-ethoxyethyl)phenyl]pyridin-3-yl}ethan-1-one
(3S,5R)-3-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine
3-({[2-(benzylsulfanyl)ethyl]carbamoyl}amino)-N,N,2-trimethylbenzamide
5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{4-ethoxy-3-[(methylamino)methyl]phenyl}benzamide
(1R,7S)-3-(2-ethoxyethyl)-6-(4-ethyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(2-aminopyridin-3-yl)methyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
1-[2-methoxy-5-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(3S,4S)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
(1-methyl-1H-imidazol-2-yl)[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]methanol
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(morpholine-4-carbonyl)piperidin-1-yl]ethan-1-one
4-[(4-fluorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(pyridin-2-yl)ethyl]acetamide
N-(2-ethylphenyl)-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
N-cyclopentyl-4-{[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}benzamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1-(2-fluorobenzoyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
(2E)-3-(4-fluorophenyl)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}prop-2-enamide
N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-[methyl({4-methyl-5-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2-methyl-4-{3-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}but-3-yn-2-ol
3-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}methyl)-6-chloro-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-2H-chromen-2-one
2-[({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]adamantan-2-ol
1-{4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one