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3-fluoro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-{[3-(difluoromethoxy)phenyl]methyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1'-(isoquinoline-5-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(3R,4S)-4-(4-methoxyphenyl)-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-amine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1-methoxypropan-2-yl)amine
1-methyl-2-[1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-1,3-benzodiazole
1-{4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-cyclopropyl-N,4-dimethylpyrimidine-5-carboxamide
(3aS,6aS)-2-acetyl-5-(1,3-benzothiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2-methylbenzenesulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(3,3,3-trifluoro-2-methylpropyl)piperidine
(3R,5S)-N-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
3-{5-[2-(methylamino)-1,3-thiazol-4-yl]-3-phenyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
9-[4-(ethylamino)pyrimidin-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(hydroxymethyl)-9-[(3-methylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]acetic acid
4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
2-{1-[(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(dimethylamino)methyl]-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
2-ethyl-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidine-5-carboxamide
1-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]methyl}piperidine-4-carboxamide
(3aR,6aS)-5-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]formamido}-N-phenylpropanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
5-{2-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}pyrrolidin-2-one
N-{2-[(2S)-2-amino-3-methoxypropanamido]-4-methylphenyl}cyclohexanecarboxamide
5,8-dimethoxy-2-(2-methoxyphenyl)-3-(morpholin-4-ylmethyl)quinoline
2,4-dimethyl-N-[4-(4-{[3-(pyridin-4-yl)propyl]amino}piperidin-1-yl)phenyl]benzamide
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-(1H-pyrazol-3-yl)piperidine
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-pyrrol-1-yl)pentan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
3-({[2-(ethylamino)pyrimidin-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
3-fluoro-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine-2-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
8-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(6-hydroxy-6-methylheptan-2-yl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-(methoxymethyl)piperidine
2-(2-chloro-4-fluorophenyl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[3-(4-fluorophenyl)phenyl]-1-(furan-3-carbonyl)piperidine-3-carboxamide
4-{4-[(5-fluoro-2-methoxyphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
(2S,4S)-4-amino-1-[2-(3-cyano-2-methyl-1H-indol-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
N-benzyl-2-(1H-imidazol-2-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
1-(3-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]urea