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(3S,9aR)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{1-[4-(methylsulfanyl)phenyl]-1H-1,2,4-triazol-5-yl}-1λ6-thiane-1,1-dione
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]piperidine-3,5-dicarboxamide
1-methyl-6-oxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,6-dihydropyridine-3-carboxamide
1-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3,3-dimethylurea
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxo-N-(propan-2-yl)acetamide
N-(furan-3-ylmethyl)-N-methyl-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
6-(2-aminoethyl)-N,2-dimethyl-N-[(3-methylpyridin-2-yl)methyl]pyrimidin-4-amine
(3R,5R)-1-(naphthalen-2-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
1-[3-(7-{[2-(hydroxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]pyrrolidin-2-one
(4S)-3-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-(2,6-dimethoxy-4-methylphenyl)-N-methylbenzamide
6-methyl-4-[3-(2-methylpropyl)pyrrolidine-1-carbonyl]-2-(pyrimidin-5-yl)quinoline
5-(4-chloro-2,6-dimethoxyphenyl)-1-methyl-1H-imidazole
1-ethyl-5-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]-2-(methylamino)pyrimidine-5-carboxamide
N-[4-(furan-2-yl)phenyl]-1-[3-(thiophen-2-yl)propanoyl]piperidine-3-carboxamide
3-ethyl-1-(2-methoxy-6-methylphenyl)-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(5-propylfuran-2-yl)methyl]-decahydro-2,7-naphthyridine-2-sulfonamide
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3-(3-methylphenyl)piperidine
1-cyclopropyl-4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyrrolidin-2-one
1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]azetidine-2-carboxylic acid
N-ethyl-N-[2-(morpholin-4-yl)ethyl]-1-benzofuran-2-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl][(4-fluoro-3-methoxyphenyl)methyl]methylamine
7-(2-methylphenyl)-4-(thiophene-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-ethylphenyl)piperidine-1-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
8-fluoro-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-(2-ethoxyethyl)-3-[(5-oxo-1,4-diazepan-1-yl)sulfonyl]benzamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxylate
2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-1,3-thiazole-4-carboxamide
4-{[(6-methylhept-5-en-2-yl)amino]methyl}-1λ6-thiane-1,1-dione
N-(1-methyl-1H-pyrazol-4-yl)-4-(pyridin-3-yloxy)piperidine-1-carboxamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4-methylpyrimidine
4-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2-oxopiperazin-1-yl)benzonitrile
1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(2,4-dimethoxyphenyl)-1-[2-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-(2-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N,1-dimethyl-N-{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-amine
2-(3,5-dimethoxyphenyl)-N-(propan-2-yl)pyridine-4-carboxamide
benzyl(methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
6-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-[methyl(4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}phenyl)amino]ethan-1-ol
2-chloro-N-[2-(pyridazine-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
N-[3-(cyclopentyloxy)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-cyclopropyl-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3,5-dimethyl-1H-indole