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4-[6-(hydroxymethyl)pyridine-2-carbonyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
5-[bis(prop-2-en-1-yl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-[4-(2-methyl-4-phenylpyridine-3-carbonyl)morpholin-3-yl]acetic acid
3-({2-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
N-(carbamoylmethyl)-2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(furan-2-carbonyl)-4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazine
3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
7-(5-methylthiophen-2-yl)-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[1-(4-acetylbenzoyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
N-(dicyclopropylmethyl)-N-methyl-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
7-cyclopentyl-2-[2-(4-fluorophenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}azetidin-3-ol
6-(2-fluoro-4-methoxyphenyl)-2-[3-(hydroxymethyl)piperidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-(2-tert-butyl-6-methylphenyl)-2-methyl-2,8-diazaspiro[4.5]decane-8-carboxamide
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-cyclopropyl-2-(4-fluorophenyl)-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}acetamide
{2-[(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)methyl]phenyl}methanol
2-(dimethyl-1,2-oxazol-4-yl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-3-{2-[(2S)-pyrrolidin-2-yl]ethyl}urea
N-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}aniline
N-[7-oxo-5-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]furan-2-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-(methoxymethyl)-N-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-({3-[2-(benzyloxy)ethyl]phenyl}methyl)acetamide
3-(2-phenylethyl)-7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1,2-dimethylpiperazine
3-(2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)pyrrolidine
2-[4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
N-ethyl-3-(3-methylpiperazine-1-carbonyl)-N-(oxan-4-yl)benzene-1-sulfonamide
1-[4-(4-fluorophenoxy)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
6-{[4-(pyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
1-methyl-5-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl](4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
3-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]quinoxalin-2-ol
ethyl 1-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)acetyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
N-tert-butyl-5-chloro-2-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[3-(pyridin-2-yl)propyl]propanamide
N-[2-(dimethylamino)ethyl]-3-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}propanamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
(3aR,6aR)-2-methanesulfonyl-5-[(5-propylfuran-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(phenoxymethyl)-1,3-oxazole-4-carboxylic acid
(1R,5S,6R)-N-[(4-phenylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide