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1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-4-[(methylsulfanyl)methyl]piperidine
1-(4-fluorophenyl)-6,6-dimethyl-N-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}morpholine-2-carboxylic acid
N-(5-methyl-1,3,4-oxadiazol-2-yl)-1-(thiophene-2-carbonyl)piperidin-3-amine
5-ethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidin-2-amine
3-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-4-[4-({[(4-chloro-2-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(1,2-oxazolidin-2-yl)pyridine-3-carboxamide
5-(1-cyclopropyl-1H-pyrrol-2-yl)-1-(2,5-dimethylphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-{[(2R,5S)-5-(quinolin-6-ylmethyl)oxolan-2-yl]methyl}piperidine-4-carboxylic acid
3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]phenol
4-[1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridine
3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
(3S,4R)-4-(4-fluorophenyl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidine-3-carboxylic acid
5-{[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-(2-methyl-1H-indol-1-yl)-N-[(3R)-oxolan-3-yl]propanamide
4-(5-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl][(4-ethylphenyl)methyl]methylamine
3-(3-fluorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-4-carboxamide
4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(oxolan-3-yl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-{1-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
N-ethyl-N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(3S,4R)-N,N-dimethyl-4-propyl-1-(quinoxalin-2-yl)pyrrolidin-3-amine
(3S,4R)-N-(4-chloro-2-methylphenyl)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carboxamide
4-(4-ethoxypiperidin-1-yl)pyrimidine-5-carboxylic acid
1-(5-fluoropyridin-3-yl)-3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
7-(3-chlorophenyl)-4-[6-(propan-2-yl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-methanesulfonamidophenyl)-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
N-methyl-2-{3-[3-(6-phenylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1-[1-(1H-imidazol-1-yl)butan-2-yl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
1-(5-{[2-(methoxymethyl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
5-{2-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[3-(2-acetylphenyl)phenyl]-2-methoxyacetamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(2S)-N-ethyl-1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)pyrrolidine-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-(1,3,4-thiadiazol-2-yl)urea
3-{5-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
4-oxo-N-[2-(propan-2-yl)phenyl]-4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}butanamide
N-(3-ethoxy-2-hydroxypropyl)-2-methyl-1-benzofuran-5-carboxamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[3-(methylsulfanyl)propanamido]pyrrolidine-2-carboxamide
N-methyl-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
(4aS,8aR)-6-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[3-(dimethylamino)propyl]-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aS,8aR)-1-(2-aminoethyl)-6-[(3,7-dimethyl-1H-indol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one