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4-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-N-methyl-1,3-thiazol-2-amine
2-(2-fluorophenyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
(4aS,8aR)-1-(3-methoxypropyl)-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
4-methoxy-N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-{[7-(but-2-ynoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-methylthiophene-2-carboxamide
[2-(1-methylpiperidin-4-yl)-3-phenylquinolin-7-yl]methanol
N-methyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-{4-methyl-3-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
5-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-2,4-dimethyl-1,3-thiazole
1-(morpholin-4-yl)-3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}propan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(thiophen-2-yl)propanamide
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]urea
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
5-(naphthalen-2-yl)-3-(3-propoxypiperidin-1-yl)-1,2,4-triazine
N-[2-(dimethylamino)ethyl]-3-{[1-(1,4-dithiepan-6-yl)piperidin-4-yl]oxy}-N-methylbenzamide
1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(3-phenoxyphenyl)methyl]acetamide
(2R,6S)-2,6-dimethyl-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}morpholine
N-benzyl-3-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)oxy]benzamide
N-[(4-methylphenyl)methyl]-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
7-(3-methoxyphenyl)-2-(4-propyl-4H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-(oxan-4-yl)piperazine-1-carboxamide
N-cyclopropyl-2-(thiophen-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
3-benzyl-4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(4-methyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]acetamide
3-benzyl-8-(9H-fluoren-2-ylmethyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-aminoethyl)-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-[(2S)-1-methylpyrrolidine-2-carbonyl]piperidine
9-methoxy-N-methyl-7-oxo-3-[(1R,2R)-2-phenylcyclopropanecarbonyl]-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2,6-difluorobenzoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
7-(3-cyclopropylpropanoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 4-[({4-[4-(oxane-4-amido)-1H-pyrazol-1-yl]phenyl}formamido)methyl]benzoate
(3aR,6aR)-2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)ethan-1-one
4-(3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-methylpyridine
N-[3-(1H-indazol-1-yl)propyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylamino)acetamide
[(3,4-dimethoxyphenyl)methyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-[(4aR,7aS)-6,6-dioxo-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-phenyl-4-(4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
2-{3-cyclopropyl-5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}pyridine
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(1H-imidazol-2-ylmethyl)acetamide
1-(4-propylpyrimidine-5-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide