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3-({4-[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
6-[({[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
N-(1,3-benzothiazol-6-yl)-2-(morpholin-3-yl)acetamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(3,4,5-trifluorophenyl)methyl]piperidine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(oxane-4-carbonyl)piperidin-3-yl]propanamide
1-(3-chloropyridin-2-yl)-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2-methylnaphthalen-1-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(3-hydroxypyridine-2-carbonyl)morpholin-3-yl]acetic acid
7-(oxan-4-yl)-2-(1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
2-(4-{[benzyl(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-cyclopropyl-2-({1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
6-(2-chlorophenyl)-2-(4-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
6-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(5-methyl-4-{[2-(morpholin-4-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperidin-3-ol
4-({3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
4-fluoro-N-{3-[4-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}benzene-1-sulfonamide
N-[(2-methoxynaphthalen-1-yl)methyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-(2-methylpropyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1,2-oxazole-5-carboxamide
4-hydroxy-2-phenyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-5-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(4-methoxy-2,3,6-trimethylbenzenesulfonyl)pyrrolidine-2-carboxamide
2-[(adamantan-1-ylmethyl)[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]amino]ethan-1-ol
N-(3-hydroxy-3-phenylpropyl)-N,1-dimethyl-5-phenyl-1H-pyrrole-2-carboxamide
N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}furan-3-carboxamide
(2R)-4-methyl-2-{[2-(pyridin-4-yl)pyrimidin-5-yl]formamido}pentanamide
2-ethyl-9-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(1-carbamoylcyclopropyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-[(5-{[3-(difluoromethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-9,10-dihydroacridin-9-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
ethyl 4-(2-methoxyethyl)-1-(2-phenylethyl)piperidine-4-carboxylate
N-(cyclohex-1-en-1-ylmethyl)-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
3-(5-chloro-2-methoxyphenyl)-1-{[4-(dimethylamino)oxan-4-yl]methyl}urea
N-{1-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}methanesulfonamide
4-(4-fluorophenyl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-4-oxobutanamide
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
2-{[4-(2,4-difluorophenyl)-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-propyl-5-{[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
3-(2-methoxyphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
3-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N,N-dimethylpropane-1-sulfonamide
(3S,4R)-1-[(4-methylphenyl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
ethyl 5-[(2,4-dimethyl-3-oxopiperazin-1-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](furan-2-ylmethyl)methylamine
2-(phenylamino)-N-[(3R)-piperidin-3-yl]pyrimidine-5-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2,3-dihydro-1-benzofuran-5-carboxamide
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(2-aminopyridine-4-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol