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N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-[2-(2,6-difluorophenyl)ethyl]piperidine
N6-benzyl-N5-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-(4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
2-{4-[(2,5-difluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(3-chloro-4-phenoxyphenyl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}oxane-4-carboxamide
5-(2-fluorophenoxymethyl)-N-[(1S)-2-hydroxy-1-phenylethyl]-1H-pyrazole-3-carboxamide
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]propanamide
N-butyl-5-(4-methanesulfonylphenyl)furan-2-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-1H-1,2,4-triazol-5-yl]morpholine
3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
ethyl 4-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-amido)piperidine-1-carboxylate
2-(2-ethoxyphenyl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
(3S,4R)-N,N-dimethyl-4-propyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-amine
N-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-3-acetamidopyrrolidine-1-carboxamide
11-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-4-(3-methylbutyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
8-(furan-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-{[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
2-{[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}-3-(furan-2-yl)propan-1-ol
4-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)azetidin-3-yl]morpholine
(4-{[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2,2-dimethyl-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]morpholine
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3,5-difluorophenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
7-chloro-4-[1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
3-(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
4-[(4-{[1-(pyridine-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]thiomorpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-ethylpyrimidine-5-carboxamide
1-[5-({[(3,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
N-[3-(3-fluorophenyl)phenyl]-1-(thiophen-2-ylmethyl)piperidine-4-carboxamide
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2R,3R)-1'-cyclopropanecarbonyl-3-(4-methylpiperazin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-fluorobenzamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}(methyl)[1-(pyridin-4-yl)ethyl]amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidine
2-[4-(quinolin-8-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(phenylsulfanyl)acetamide
1-(2-methyl-5-propylpyrimidin-4-yl)-N-(oxan-4-yl)piperidin-4-amine
2-(ethylamino)-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]pyrimidine-5-carboxamide
1-(4-benzylpiperazin-1-yl)-3-(1-cyclopropanecarbonylpiperidin-3-yl)propan-1-one
2-[1-(furan-3-ylmethyl)-4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-2-yl]ethan-1-ol
1-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine