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{1-[2-(2,5-difluorophenyl)ethyl]piperidin-2-yl}methanol
5-[phenyl({[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino})methyl]-1,3,4-thiadiazol-2-amine
4-[2-(4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]morpholine
(4S)-N-[(4-fluorophenyl)methyl]-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
1-(3-chloro-4-methoxyphenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(oxolane-2-carbonyl)piperidin-4-yl]oxy}benzamide
7-chloro-4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-5-propyl-1,2-oxazole-3-carboxamide
methyl 3-cyclopropaneamido-6-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
1-[(4-methylphenyl)methyl]-4-[2-(2,3,4-trifluorophenyl)acetyl]piperazin-2-one
(3S,4S)-4-(propan-2-yl)-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxylic acid
N'-[2-(4-chlorophenyl)ethyl]-N-(2-ethoxyphenyl)propanediamide
(3S,4R)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidin-4-amine
3-hydroxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4-methylbenzamide
ethyl 1-(3-hydroxybutyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[(3,4-difluorophenyl)methyl]-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}propanamide
1-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(2-methylphenyl)-1H-imidazole
N-[cyclohexyl(thiophen-2-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
3-(2,6-dimethylphenoxy)-1-(furan-3-ylmethyl)azetidine
1-(6-chloropyridin-3-yl)-3-{pyrazolo[1,5-a]pyridin-3-ylmethyl}urea
(2S,4S,5R)-1-methyl-2-(2-methylpropyl)-4-(morpholine-4-carbonyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-cyclohexyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
10-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
4-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-(3-fluorophenoxy)-1-[2-(3-methyl-1,2-oxazol-5-yl)ethyl]piperidine
N-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylthian-4-amine
5-(1,4-dimethyl-1H-indazol-3-yl)pyridin-3-amine
3-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
4-[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octane-3-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-(morpholin-4-yl)-N-[(1-phenylcyclopentyl)methyl]benzamide
4-[(dimethylamino)methyl]-4-hydroxy-N-(4-phenylphenyl)azepane-1-carboxamide
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
4-[(2,3-difluorophenyl)methyl]-3-[2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
2-tert-butyl-N-[2-(3-chlorophenyl)ethyl]-4-hydroxypyrimidine-5-carboxamide
1-methyl-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3-(5-propyl-4H-1,2,4-triazol-3-yl)urea
2-amino-4-(furan-2-yl)-6-(3-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N,1-dimethyl-6-oxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,6-dihydropyridine-3-carboxamide
2-(cyclopropylmethyl)-7-(4-hydroxy-2-methylpyrimidine-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2-methyl-3-{[(2-phenoxyethyl)amino]methyl}-1H-indol-1-yl)acetamide
1-{[4-(difluoromethoxy)phenyl]methyl}-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-{4-[1-(2-methoxyethyl)-6-oxopiperidine-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
3-{[(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)amino]methyl}piperidin-3-ol
N-[2-(dimethylamino)ethyl]-3-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-yl)propanamide
3-[(dimethylamino)methyl]-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-ol
2-methoxy-1-{1'-[2-(morpholin-4-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}-N-[1-(thiophen-3-yl)propan-2-yl]acetamide