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2-[N-(1-methylpiperidin-4-yl)-1-(3,5,7-trimethyl-1H-indol-2-yl)formamido]acetic acid
2-methanesulfonyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
3-(1H-indol-3-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
1-[(3-methylpyridin-2-yl)methyl]-4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
3-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
3-(3-methoxyphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
4-fluorophenyl (7S,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-8-(3,3,3-trifluoropropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(6-methylpyridin-2-yl)methyl]-2-(3-phenylpropyl)morpholine
4-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
1-{[({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)carbamoyl]methyl}piperidine-4-carboxamide
3-benzyl-1-methyl-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(methylamino)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyridine-3-carboxamide
ethyl 4-[6-(2-cyclopentyl-2-phenylacetyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-methylphenol
1-methyl-4-(4-oxo-4H-chromen-3-yl)-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopropyl-N-{[3-(2-methylpropoxy)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-chloro-6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}pyridine-2-carboxylic acid
4-{1-cyclohexyl-5-[5-(hydroxymethyl)furan-2-yl]-1H-1,2,4-triazol-3-yl}benzamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
1-(4-{[(cyclopropylmethyl)(methyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
4-(2,4-difluoro-3-methoxyphenyl)-1-[(2S)-oxolan-2-ylmethyl]-1H-1,2,3-triazole
N-(2-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenoxy}ethyl)acetamide
3-(4-fluorophenyl)-4-(piperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(4-chloro-1H-pyrazol-1-yl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}propanamide
4-(1H-imidazol-2-yl)-1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]piperidine
1-(azepan-1-yl)-3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)-6-methylpyridine
4-(1-{1-[3-(1H-imidazol-1-yl)propyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
3-benzyl-4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
1-(2-chlorobenzoyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
2-{2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4R)-4-amino-1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
8-(2-acetylbenzoyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
3-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-methyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3S,4S)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
1-{2-[1-cyclohexyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
4-phenyl-N-{[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]methyl}benzamide
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
(1S,5R)-3-(3-methoxypropyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3-fluorophenyl)methyl]-N-methyl-6-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
[5-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)furan-2-yl]methanol
(2S,4R)-N,N-diethyl-4-(6-methyl-4-oxo-4H-pyran-2-amido)-1-propylpyrrolidine-2-carboxamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2,3,4-trimethoxybenzamide
2-phenyl-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine