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6-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
1-[1-methyl-5-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}piperidin-2-one
N-(1-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
N-[4-(furan-2-yl)butan-2-yl]-3-phenyl-1H-pyrazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}furan-2-carboxamide
1-(2-methylphenyl)-4-(piperidin-3-yl)piperazine
3-[2-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
4-{6-[3-(pyridine-3-carbonyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
(4aS,8aR)-6-(5-hydroxypyrazine-2-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-ethoxy-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-(4-methoxy-2-methylphenyl)acetamide
methyl (2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-(4-fluorobenzamido)pyrrolidine-2-carboxylate
(1R,5R)-6-[2-(2-ethylphenoxy)ethyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-[2-(2-ethylphenoxy)ethyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyrrolidin-3-yl)benzamide
8-fluoro-N-[1-(4-fluorophenyl)-2-hydroxyethyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
3-(3-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-1H-indol-1-yl)propanamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
5-[(furan-2-ylmethyl)amino]-1-methyl-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(thiophen-2-yl)butanamide
2-[3-(propan-2-yl)-5-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,4-triazol-1-yl]pyridine
5-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2-fluoro-4-methylphenyl)-2-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]acetamide
3-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanamide
[(2-butyl-1H-imidazol-4-yl)methyl]({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
(4S)-3-[2-(azepan-1-yl)-2-oxoethyl]-4-phenyl-1,3-oxazolidin-2-one
N-(1-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
8-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
3-{2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-oxoethyl}-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-{[1-(dimethylamino)cyclohexyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-(3-hydroxypyridine-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-(dimethylamino)-N-[(2,6-dimethylpyridin-4-yl)methyl]-2-(4-methylphenyl)acetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
7,7-dimethyl-2-(5-phenyl-4H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
4-(4-{[(2-benzyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
2-(2-methoxyethyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,3-benzoxazole-6-carboxamide
6-chloro-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
(3aS,7aR)-5-methyl-2-(2-propyl-1,3-thiazole-4-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
N-(8-chloroquinolin-5-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2-methoxy-1-{1'-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one