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4-(1H-imidazol-2-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
(5S)-5-{[({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(pyridin-2-ylmethyl)amino]methyl}pyrrolidin-2-one
N-(1-methyl-1H-pyrazol-4-yl)-2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
2-{2-[(1-methylpiperidin-4-yl)methyl]pyrimidin-4-yl}pyridine-4-carboxylic acid
5-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclopropane-1-carboxamide
N-(1,2-oxazol-3-ylmethyl)-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
N-(2-{7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-ethyl-4-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydropyridin-2-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
4-(2-methylpyrrolidine-1-carbonyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
6-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(2S)-2-acetamido-N-[2-(2-ethylphenoxy)ethyl]-N-methylpropanamide
2-methyl-4-(4-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenyl)butan-2-ol
(2R,3R,6R)-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-benzyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)piperazin-2-one
N-methyl-N-(2-methylprop-2-en-1-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanamido]-N-(2-ethylphenyl)benzamide
2-propyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyridine-4-carboxamide
5-[(cyclobutylamino)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(cyclopropylmethyl)-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2-(propan-2-yl)-1,4-diazepane
(1R,3S)-7-[(5-chloro-2,3-dimethoxyphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-benzothiophene-5-carboxamide
4-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanamide
N-[(3-fluorophenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
2-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-5-methylpyrazine
(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-(oxane-4-carbonyl)-8-azabicyclo[3.2.1]octane
4-(2-ethylphenyl)-3-(1-methyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-methoxy-5-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
[(4aS,8aR)-1-(cyclopentylmethyl)-6-(pyrazine-2-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
1-[(2,5-difluorophenyl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
1-(6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}pyrimidin-4-yl)piperidin-4-ol
7-[(3,4-difluorophenyl)methyl]-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
1-(5,6-dimethylpyridine-3-carbonyl)-4-[3-(4-fluorophenoxy)propyl]piperazine
(1,4-dioxan-2-ylmethyl)[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
5-{1-[(2,5-dimethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
ethyl (4aS,8aR)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylate
2-(2-{[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
5-[(3-ethoxy-4-methoxyphenyl)methyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
4-[(5-ethylfuran-2-yl)methyl]-2-(2-methoxyethyl)morpholine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)quinoline-4-carboxamide
(2-{1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)dimethylamine