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3-[(2-methoxyethyl)(pyridin-4-ylmethyl)sulfamoyl]-N,N-dimethylbenzamide
7-(5-methylthiophen-2-yl)-4-(piperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-methoxyethyl)-8-[(3-methoxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-butanamido-3-methoxyphenyl)-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
methyl 1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
[(3R,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(dimethylamino)ethyl]-3-[1-(propane-1-sulfonyl)piperidin-4-yl]propanamide
1-[bis(4-fluorophenyl)methyl]-4-[(2R)-pyrrolidine-2-carbonyl]piperazine
2-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
2-benzyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1,3-thiazole-4-carboxamide
[(2-methyl-2H-indazol-3-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
N-ethyl-N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-(1-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxypyridine
5-{4-phenyl-1-[2-(pyridin-3-yloxy)propyl]-1H-imidazol-5-yl}pyrimidin-2-amine
2-[2-(1H-indazol-1-yl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-[1-(1-benzylpyrrolidin-3-yl)-1H-1,2,3-triazol-4-yl]pyrimidine
N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}propanamide
2-(2-chloro-4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
4-(benzyloxy)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-[4-(furan-2-yl)phenyl]-3-[2-(propane-2-sulfonyl)ethyl]urea
N,8-dimethyl-N-(2-phenylethyl)-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
8-(2-amino-6-methylpyrimidin-4-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-methoxyphenyl)acetamide
(3S,4R)-1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-3-methoxypiperidin-4-amine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)ethyl]pyridine-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
4-{4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
4-[ethyl(5-phenylpentyl)amino]butan-1-ol
(3S,4R)-1-(1H-indazole-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
2-(2-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
3,5-dimethoxy-N-({1-[3-(1-methylcyclopropyl)propanoyl]piperidin-3-yl}methyl)benzamide
4-(isoquinolin-1-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,4S)-N-[3-(cyclopentyloxy)phenyl]-4-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carboxamide
2-(2-oxo-1,3-oxazolidin-3-yl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]acetamide
N-[(3-chlorophenyl)methyl]-4-acetamido-N-propylbutanamide
3-(3-methylbutyl)-8-[2-(1H-pyrazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{3-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
1-{1-[(4-methanesulfonylphenyl)methyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
3-(2-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
4-(2-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)morpholine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(dimethyl-1,2-oxazole-4-carbonyl)pyrrolidine-3-carboxylic acid
5-(2-chlorophenyl)-4-[1-(cyclohex-3-en-1-ylmethyl)piperidin-3-yl]pyrimidine
[2-(1H-imidazol-1-yl)ethyl](methyl){[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine