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1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
4-[2-(4-methoxyphenoxy)acetyl]-1-(2-methylphenyl)piperazin-2-one
methyl 1-{3-[(2-hydroxyethyl)amino]-5-(pyrrolidine-1-sulfonyl)benzoyl}piperidine-2-carboxylate
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}amine
1-[(3-fluorophenyl)methyl]-4-(6-methoxypyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2R,3R)-3-amino-1'-[(5-methylnaphthalen-1-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
7,7-dimethyl-2-(3-methylphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-ethoxypropyl)acetamide
1-{4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(5-methylfuran-2-yl)methyl]amine
8-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-(4-cyano-2-fluorophenyl)azocane-1-carboxamide
(butan-2-yl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})(pyridin-3-ylmethyl)amine
6-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
6-(difluoromethyl)-2-(3-{[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-{3-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]propanamido}benzamide
[(2S,4R)-1-(2,5-dimethoxybenzenesulfonyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N'-(2-ethoxyphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanediamide
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(2S,4S)-N-ethyl-4-[2-(thiophen-3-yl)acetamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
3-methyl-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
2-phenoxy-N-(1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
1-({5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
4-ethyl-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-4-cyclohexanecarbonylpiperazine-1-sulfonamide
2-[1-(3-methylphenyl)-1H-pyrazol-3-yl]pyrazine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)but-2-ynamide
(3S,4R)-4-(hydroxymethyl)-1-[(4-methoxy-5,6,7,8-tetrahydronaphthalen-1-yl)sulfonyl]piperidin-3-ol
2-({6-[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
1-butyl-5-(2-fluoro-6-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
4-methyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]piperidine-4-carboxamide
2-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]-1,3-benzoxazole
N-cyclopropyl-1-(8-fluoro-4-oxo-1,4-dihydroquinoline-2-carbonyl)piperazine-2-carboxamide
4-[(6-cyclopropylpyrimidin-4-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
5-(2-methoxy-4-methylphenoxymethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-(2-chlorophenyl)piperidine-1-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
1-(4-fluorophenyl)-4-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]butan-1-one
{2-[(2,1,3-benzoxadiazol-5-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl}dimethylamine
(3S,4R)-3-benzyl-1-(2,6-diaminopyrimidin-4-yl)-4-methylpiperidin-4-ol
5-methanesulfonyl-N-(naphthalen-1-ylmethyl)-4-(piperidin-3-yl)pyrimidin-2-amine
8-fluoro-2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]quinoline