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2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-ethyl-5-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyrimidin-2-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-2-one
4-tert-butyl-N-(oxolan-3-yl)benzamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-4-(piperidin-1-yl)butanamide
methyl 8-[(3-chlorophenyl)methyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
4-(4-{[1-(2-methoxyphenoxy)propan-2-yl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
N-benzyl-N,1-dimethyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(morpholin-3-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
(3aR,6aR)-2-cyclopropanecarbonyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-chloro-4-fluoro-N-(1,2-oxazol-3-ylmethyl)-1-benzothiophene-2-carboxamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
3-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
(4aR,8aR)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
7-methyl-4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}thieno[3,2-d]pyrimidine
2-(1H-indol-3-yl)-1-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-(2-cycloheptylethyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-[3-(1H-indol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N,N-dimethyl-6-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridazin-3-amine
2-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}quinoline
N-[(3R,5S)-1-cyclohexyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
N-cyclopropyl-2-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
4-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-5-fluoroquinazoline
1,3-dimethyl-2,6-dioxo-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-acetyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]thiophene-3-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-5-one
N-[(1-benzylpiperidin-4-yl)methyl]-N,2-dimethylpyridin-4-amine
(5S,9aS,9bS)-5-(2-chlorophenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
methyl 3-{[5-(methoxymethyl)furan-2-yl]methyl}-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
5-(4-chlorophenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-{[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyrrolidin-3-ol
N-[2-(methylsulfanyl)phenyl]-N'-(oxan-2-ylmethyl)butanediamide
4-methyl-2-(pyridin-3-yl)-5-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrimidine
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-amino-4-(2,1,3-benzoxadiazol-4-yl)-6-cyclopropanecarbonyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N'-(5-chloro-2-methylphenyl)-N-(1-methanesulfonylpiperidin-4-yl)propanediamide
N-[(2R,3R)-1'-(1-methylcyclopropanecarbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-(2-ethylbutyl)-8-(oxolane-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]pyrimidine-5-carboxamide
5-tert-butyl-1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N4-[(2,3-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-(methylsulfanyl)-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide