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(3aR,6aR)-2-(prop-2-en-1-yl)-5-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(5-fluoro-2-methylphenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-benzyl-3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-methylpropanamide
4-(2-methylquinolin-6-yl)-1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-ol
5-fluoro-N4,N4-dimethyl-N2-[1-(oxan-4-yl)piperidin-4-yl]pyrimidine-2,4-diamine
2-(5-fluoro-2-methylphenyl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
N-[3-(1H-indol-1-yl)propyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
(3aR,6aR)-2-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)sulfamoyl](ethyl)methylamine
6-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1,4-oxazepan-6-ol
[2-(7-methyl-1H-indol-3-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
8-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
ethyl 3-{[5-(2,6-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-5-methylhexanoate
[2-({4-[(3,5-dichlorophenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-[(3S,4R)-1-{2-[4-(dimethylamino)phenyl]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-(2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-4-phenylphenoxy)acetamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
6-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}pyridine-2-carbonitrile
1-[4-(furan-2-carbonyl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-[2-(2,3-dimethylphenoxy)ethyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-4-cyclopropyl-1-(pyrazin-2-yl)pyrrolidin-3-yl]-2-methanesulfonamidoacetamide
3-methyl-6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridazine
N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(naphthalen-1-ylmethyl)butanamide
N-[2-(3-methoxyphenyl)-1-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
1-{1'-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
4-chloro-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
5-{2-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-(2-methyl-1H-imidazol-1-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-(2-hydroxyethyl)piperidine-4-carboxamide
N-[3-(cyclopentyloxy)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-acetamido-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
3-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
4-(2-fluoro-3-methoxyphenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
2-{4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperazin-1-yl}-1,3-benzoxazole
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
4-(4-{[(2R,6S)-2,6-dimethylpiperidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)-N-[(2R)-3-methylbutan-2-yl]piperidine-1-carboxamide
N,N-dimethyl-7-(propane-1-sulfonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(dimethylamino)-N-[(1-ethylcyclobutyl)methyl]-2-(2-methylphenyl)acetamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(pyridin-4-yl)pyrimidin-2-amine
methyl 3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-methoxypyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
N-(2-methoxyethyl)-1-methyl-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
N-[(3,4-dimethoxyphenyl)methyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
N,6-dimethyl-2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine