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N,N-diethyl-1-{2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetyl}piperidine-4-carboxamide
(3aR,6aR)-2-acetyl-5-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-4-methoxyphenol
N-[(1-methylpiperidin-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
(3S,4R)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2,4-dimethoxy-5-[4-(1-methoxyethyl)phenyl]pyrimidine
N-[(2R,3R)-1'-[(5-chloro-2-hydroxyphenyl)methyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
7,11-dimethyl-N-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3,7,11-triazaspiro[5.6]dodecane-3-carboxamide
2-(3-hydroxyphenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
2-[2-(2-fluoro-5-methoxyphenyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
N4,N4,N6-trimethyl-N6-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-4,6-diamine
1-{4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]thiophen-2-yl}ethan-1-one
11-[bis(prop-2-en-1-yl)amino]-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 5-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-(pyrrolidine-1-carbonyl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperidine
(benzylsulfamoyl)({[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl})amine
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylacetamide
1-{4-[2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}pent-4-en-1-one
N-(2-methyl-4-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]carbamoyl}phenyl)furan-2-carboxamide
(3R,4S)-4-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
N,2,5-trimethyl-1-phenyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrole-3-carboxamide
N-(2-methoxyethyl)-2-(pyrrolidin-3-yl)-N-(thiophen-2-ylmethyl)acetamide
8-[6-(methoxymethyl)pyrimidin-4-yl]-1-oxa-8-azaspiro[4.5]decan-3-ol
2-cyclopentyl-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
3-ethyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
(3S,4R)-4-methyl-1-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}piperidine-3,4-diol
4-(2,6-dimethylpyridin-3-yl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrimidin-2-amine
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
2-(4-fluorophenoxymethyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-3-carboxamide
N-cyclopentyl-1-(2-methylpropyl)-5-(1,2,3-thiadiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
2-[cyclopentyl(methyl)amino]-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]ethan-1-one
1-cyclopropanecarbonyl-N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxamide
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2,2-dimethylpropanoyl)pyrrolidin-3-yl]-4-(1H-pyrazol-4-yl)butanamide
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}[(4-methyl-1H-imidazol-2-yl)methyl]amine
8-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 2-[3-(3-chlorophenyl)-3-(3-hydroxyphenyl)propanamido]acetate
7-cyclohexyl-2-(2-hydroxy-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
5-[(4-methanesulfonylphenyl)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-(2-hydroxyethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]azocane
1-(2-phenylethyl)-4-[3-(pyridin-2-yl)propanoyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-(2-aminoethyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-4-ethyl-1-{2-[(2-phenylethyl)sulfanyl]pyridine-3-carbonyl}piperidine-3,4-diol
methyl 1-{3-[(2-ethoxyphenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
6-{4-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}pyridine-3-carboxamide
3-(4-methoxyphenyl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
1,5-dimethyl-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1H-indazole