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5-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxylic acid
1-(carbamoylmethyl)-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]piperidine-4-carboxamide
N-methyl-5-(1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(oxolan-2-ylmethyl)-9-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
(2R,3R,6R)-5-(1H-1,2,3-benzotriazole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-5-methoxy-1-methyl-N-[2-(phenylsulfanyl)ethyl]-1H-indole-2-carboxamide
N-[3-(aminomethyl)phenyl]-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
(2E)-1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
5-[4-(3-chlorophenyl)piperazin-1-yl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
3-{4-[(2-butyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}-6-chloropyridazine
5-ethyl-2-{1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazol-2-yl}pyridine
3-{2-[6-(dimethylcarbamoyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}propanoic acid
5-(3-phenylpiperazine-1-carbonyl)-4-propylpyrimidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetamide
(4aR,7aS)-1-{2-[methyl(1H-pyrazol-3-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-methyl-14-(3-phenoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-benzyl-1-methyl-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
4-[3-(2-methoxyethyl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl]-1-methyl-1,2-dihydroquinolin-2-one
3-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2,6-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidine-4-carboxamide
(3R,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({4-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}methyl)-2-methylpropanamide
(1R,7S)-6-(4-methyl-1,4-diazepane-1-carbonyl)-3-(3-methylbutyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]pyridin-2-amine
(2S)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1H-imidazol-4-yl)propanamide
2,6-dimethyl-4-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]quinoline
5-(3-methoxyphenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-{1-[1-(ethanesulfonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
1-[4-(hydroxymethyl)benzoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-3,3-dimethylurea
2-methyl-4-(5-{[propyl(pyridin-3-ylmethyl)amino]methyl}thiophen-2-yl)but-3-yn-2-ol
1-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-2-ethyl-5-fluoro-1H-1,3-benzodiazole
1-cyclopentyl-N-ethyl-5-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-({8-[(3-ethoxy-4-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
2-{4-[(2-methylnaphthalen-1-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-methyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
3-[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]-N-(3-methylphenyl)propanamide
N-(3-hydroxy-3-phenylpropyl)-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-methylpropanamide
3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)phenol
4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
6-[(2-methoxyphenyl)methyl]-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-cyclopropyl-2,8-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]quinoline-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide