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11-{[(2,3-difluorophenyl)methyl]amino}-4-[2-(pyridin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-5-(propan-2-yl)pyrimidin-4-amine
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
N-(2-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
5-(3-methoxyphenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-3-(1H-pyrazol-1-yl)benzamide
[(4-methyl-1H-imidazol-2-yl)methyl]({[2-(2-methylpropoxy)-7-(methylsulfanyl)quinolin-3-yl]methyl})amine
1-[2-(4-ethoxypiperidin-1-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
2-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,2,3,4-tetrahydroisoquinoline
3-methyl-6-[5-(2,2,3,3-tetramethylcyclopropyl)-1,2,4-oxadiazol-3-yl]pyridazine
2-(morpholin-4-ylmethyl)-1H-1,3-benzodiazole
1-(2,3-dihydro-1H-inden-2-yl)-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
2-(1-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole
N-[(3S,4R)-1-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(2-ethoxyethyl)-N-[2-(5-methylfuran-2-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(2-methyl-1H-imidazol-1-yl)propanamide
1-(furan-3-carbonyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
2-[(1-acetylpiperidin-4-yl)oxy]-N-cyclohexyl-5-methoxybenzamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
N-[3-({[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamoyl}methoxy)phenyl]propanamide
N-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}methanesulfonamide
dimethyl(2-{[5-(pyrrolidine-1-carbonyl)furan-2-yl]oxy}hex-5-en-1-yl)amine
2-(2H-1,3-benzodioxol-5-yl)-5-(furan-3-ylmethyl)-8-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-{4-[(trifluoromethyl)sulfanyl]phenyl}pyrrolidine-1-carboxamide
1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-phenoxybutan-1-one
4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
(2R)-N-(1H-1,2,3-benzotriazol-4-yl)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}propanamide
3-(2-ethyl-1H-imidazol-1-yl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
3-{5-[(2,4-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[3-(piperidin-1-yl)azetidin-1-yl]ethan-1-one
N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]-N-(1H-pyrazol-3-ylmethyl)pyrrolidine-3-carboxamide
4-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(2S)-2-[(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazol-4-yl)formamido]-4-methylpentanamide
methyl (2S,4S)-1-[(3-chlorophenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(1H-1,3-benzodiazol-1-yl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
N,1,6-trimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-(carbamoylmethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 1-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylate
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-(2-methoxyacetyl)-N-{3-[(pyridin-3-yl)amino]propyl}piperidine-3-carboxamide
2-methyl-5-[4-(pyrrolidin-3-yl)piperazine-1-carbonyl]phenol
4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine