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1-{3-[(4-fluorophenyl)methoxy]azetidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[4-(3-fluorophenyl)phenyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-3-carboxamide
(1S,5R)-6-[(3,5-dimethoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-3-phenoxypropanamide
3-ethyl-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
4,6-dimethyl-2-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-3-carbonitrile
methyl 6-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]pyrimidine-4-carboxylate
1-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
4-{1-[4-(furan-2-yl)benzoyl]piperidin-3-yl}-5-methyl-2-(pyridin-3-yl)pyrimidine
{[4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
3-(carbamoylmethoxy)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)benzamide
5-methyl-N-[2-(morpholin-4-yl)ethyl]-2-phenyl-1H-imidazole-4-carboxamide
2-{4-[(2,4-dimethylphenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
N-(4-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}phenyl)acetamide
N5-tert-butyl-N3-cyclohexyl-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-N-[(4-phenoxyphenyl)methyl]-1-propyl-1H-pyrazole-5-carboxamide
({4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine
1-cyclohexyl-4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1,4-diazepane
methyl 2-{8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
3-fluoro-4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
ethyl 2-({3-[(1H-indol-2-ylformamido)methyl]piperidine-1-carbonyl}amino)acetate
(3S)-3-({5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)azepan-2-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine
1-(2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)piperidin-3-ol
3-methoxy-N-[1-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-6-methyl-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-propylpiperidine-3-carboxylic acid
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(propan-2-ylsulfanyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(4-fluorophenyl)propyl]-1,4-oxazepane
4-(2-methyl-1H-imidazol-1-yl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
4-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinazolin-2-one
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
N-[(2-chlorophenyl)methyl]-4-(2-oxopyrrolidin-1-yl)-N-(prop-2-en-1-yl)benzamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-4H-chromen-4-one
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
2-(3-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[3-(4-fluorophenyl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
propan-2-yl 4-chloro-3-{[(1S,5S)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]amino}benzoate
1-methyl-2-(morpholin-4-yl)-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
(3S,7S,8aS)-3-(4-aminobutyl)-7-(benzylamino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
[(1-cyclopentylpiperidin-4-yl)methyl]({[4-methoxy-3-(methoxymethyl)phenyl]methyl})(pyridin-3-ylmethyl)amine
2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}-N-(1,3-thiazol-2-yl)acetamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-{1-[(1-ethyl-1H-indol-6-yl)methyl]piperidin-4-yl}methanesulfonamide