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4-(4-methyl-1H-pyrazol-1-yl)-1-{[4-(pyridin-2-yl)phenyl]methyl}piperidine-4-carboxylic acid
{1-[(4-fluorophenyl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
(2-chlorophenyl)(3-cyclopentyl-1-methyl-1H-1,2,4-triazol-5-yl)methanol
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclobutanecarboxamide
N-[2-(2-methylphenoxy)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-methyl-4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,5-dimethoxybenzene-1-sulfonamide
1-[4-(morpholin-4-yl)benzoyl]-1,4-diazepan-6-ol
7-(2,2-dimethylpropyl)-2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methanol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(morpholine-4-carbonyl)piperidine-4-carboxylic acid
N3-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]piperidine-1,3-dicarboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-(oxolane-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(morpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]piperidin-2-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
methyl N-{2-oxo-2-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}carbamate
8-fluoro-4-oxo-N-(2,2,2-trifluoroethyl)-1,4-dihydroquinoline-2-carboxamide
2-(2,5-dimethylphenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
5-methyl-2-(5-methylthiophen-2-yl)-4-[2-(pyrrolidine-1-carbonyl)phenoxymethyl]-1,3-oxazole
2-hydroxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyridine-3-carboxamide
5-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine-2,4-diol
4-{1-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]ethyl}morpholine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(1H-imidazol-4-ylmethyl)(oxolan-2-ylmethyl)amine
4-[6-(methoxymethyl)pyrimidin-4-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-butyl-4-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-1-methylpiperazin-2-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
3-(but-2-yn-1-yl)-5-(1-{[4-(dimethylamino)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
2-chloro-N-[1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)propan-2-yl]pyridine-4-carboxamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
methyl 2-(morpholine-4-sulfonyl)-6-{[4-(propan-2-yl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[2-(pyridin-3-yloxy)propyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
[(3S,4S)-4-(hydroxymethyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]methanol
4-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
7-(2,1,3-benzothiadiazol-5-ylmethyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-1,2,3-triazol-4-yl}-6-methylpyridine
3-ethyl-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}piperidine-3-carboxylic acid
N-[(1,1-dioxo-1λ6-thian-4-yl)methyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
methyl 3-{[2-(1H-1,3-benzodiazol-1-ylmethyl)-1,3-oxazol-4-yl]formamido}propanoate
N-{2-[1-(4-methylpyridin-2-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-[3-(1H-indol-2-yl)phenyl]-1-(oxan-4-yl)piperidine-3-carboxamide
methyl 3-[(4-methyl-1H-imidazol-5-yl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
2-(dimethylamino)-4-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]pyrimidine-5-carboxamide
3-(1-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
6-(4-hydroxyphenyl)-2-methyl-3,4-dihydroquinazolin-4-one