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(2S)-3-phenyl-2-[(3-propyl-1H-pyrazol-5-yl)formamido]propanamide
2-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
3-{[(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
3,5,7-trimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-1H-indole-2-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
9-hydroxy-3-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-(2-ethoxyethyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-2-(2,2-dimethyloxan-4-yl)-1H-imidazole
(2E)-3-(4-methoxyphenyl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
3-ethyl-8-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4S,5R)-1-methyl-2-(2-methylpropyl)-4-[(2-methylpropyl)carbamoyl]-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
(3R,4R)-3-cyclobutyl-4-methyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-methyl-N-(1-methylpyrrolidin-3-yl)acetamide
6-{2,8-diazaspiro[4.5]decan-2-yl}-9H-purin-2-amine
1-cyclohexyl-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-(1H-indole-2-carbonyl)-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1,4-dioxane-2-carboxamide
3-[(2-methoxyethyl)sulfamoyl]-5-{pyrazolo[1,5-a]pyridin-7-yl}benzoic acid
5-({2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-3-(propan-2-yl)-1,2-oxazole
1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azonane
N-cyclohexyl-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
3-[(dimethylamino)methyl]-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-ol
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
N-[(1-benzylpiperidin-4-yl)methyl]-5-(1H-imidazol-1-ylmethyl)-N-methylpyridin-2-amine
3,5-dimethyl-1-(2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}ethyl)-1H-pyrazole
4-{5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}-1-methylpiperidine
N-methyl-3-(5-methylfuran-2-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
2-(5-{1-[(2S)-2-methoxy-2-phenylacetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
ethyl (4aS,8aR)-6-[(2-methyl-1,3-thiazol-4-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylate
6-[(1-propylcyclobutyl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-{1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propanoic acid
[2-(1-methylpyrrolidin-2-yl)ethyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
2-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,3-dihydro-1H-isoindole
8-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
7-cyclohexyl-N-(2-fluorophenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(3R,4R)-1-(2-ethylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
3-[3-(2-methoxyethyl)-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
1-(4-benzylpiperidin-1-yl)-3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propan-1-one
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)pyridine-2-carboxamide
2-(dimethylamino)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-methylpyrimidine-5-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
5-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepan-6-yl]oxy}acetamide
N-[4-(furan-2-yl)phenyl]-1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidine-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-4-(piperidin-1-ylmethyl)benzamide
3-cyclopentyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]propanamide