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2-(ethylamino)-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}phenol
5-{3-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methoxyphenyl)methyl]pyrrolidin-2-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
4-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methylpyridine
1-(cyclohexylmethyl)-2-(methoxymethyl)-6-methyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-(4-chloro-2-fluorophenyl)-2-{[3-(pyridin-3-yl)propyl]amino}acetamide
4-{1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}-1,4-diazepan-2-one
(1R,5S)-3-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-3,8-diazabicyclo[3.2.1]octane
8-(3,3-dimethylbutanoyl)-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(furan-2-yl)propan-1-one
N-methyl-2-(methylsulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-methoxybutyl)-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
1-[2-(4-methoxyphenyl)ethyl]-4-({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amino)pyrrolidin-2-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(cyclohexylmethyl)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-methyl-2-({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)acetamide
2-(thiophen-3-ylmethyl)-4-{4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(furan-2-ylmethyl)-4-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]pyridine-2-carboxamide
N3,N3-dimethyl-N5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,4-thiadiazole-3,5-diamine
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxylate
2-{11-oxo-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1(9),2,4,7-tetraen-5-yl}benzonitrile
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4S)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-cyclopropyl-1-(oxan-4-yl)-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
4-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
methyl (2S,4R)-1-[(4-chlorophenyl)methyl]-4-(3-hydroxynaphthalene-2-amido)pyrrolidine-2-carboxylate
2-(2-aminoethyl)-N-[1-(4-methylpyridin-2-yl)propyl]quinazolin-4-amine
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(2-ethylphenoxy)ethyl]-N-methylacetamide
4-(carbamoylmethyl)-N-[3,5-difluoro-4-(trifluoromethyl)phenyl]piperazine-1-carboxamide
N-[3-(4-methylpiperazin-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-methyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3-(2-oxoimidazolidin-1-yl)benzamide
4-(1H-imidazol-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carbonitrile
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(4-butyl-2,3-dioxopiperazin-1-yl)-2-phenylacetamide
5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
2-methoxyethyl 4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-(2-methoxyethyl)-5-[(2S)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
(2S)-2-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-hydroxypropan-1-one
5-methoxy-9-(pyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecane