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3-benzyl-1-(5-methyl-1H-indazole-3-carbonyl)piperidine-3-carboxylic acid
2-[3-(2-methoxyquinolin-3-yl)phenoxy]propanamide
2-[(4-chlorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-{1-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
5-(2-chlorophenyl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]furan-2-carboxamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,3-dimethyl-1H-pyrazole-5-carboxamide
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)pyridine-2-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
4-(morpholin-4-yl)-6-[4-(pyrimidin-2-yloxy)piperidin-1-yl]pyrimidin-2-amine
methyl 3-({1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}carbamoyl)propanoate
N4-methyl-N2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
3-(1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-3-yl)propanamide
3-(2-chlorophenyl)-6-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-3-methoxypyrazine
3-methyl-3-[3-(oxolan-2-yl)propyl]-1-[3-(1H-pyrazol-5-yl)phenyl]urea
2-[(4-methoxyphenyl)methyl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(2S,4R)-4-{4-[2-(furan-2-ylformamido)propan-2-yl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
4-propyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrimidine
2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)-N-(propan-2-yl)acetamide
3-phenyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(4H-1,2,4-triazol-4-yl)benzamide
3-amino-N-{[1-(pentan-3-yl)piperidin-4-yl]methyl}benzamide
6-{3-[4-(diphenylmethyl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
6-cyclopentyl-N,1-dimethyl-N-[3-(oxolan-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-{4-[1-(N-methyl-1-pyridin-2-ylformamido)-2-phenylethyl]piperidine-1-carbonyl}benzoate
ethyl 1-[1-(methylsulfanyl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)(pyridin-3-ylmethyl)amine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N3-(butan-2-yl)-1-cyclopentyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-[(3-fluorophenyl)methyl]-6-oxo-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methyl-3-(1H-pyrrol-1-yl)benzamide
ethyl (4aS,8aR)-6-(furan-3-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-4-ethenylbenzamide
[(2-butyl-1H-imidazol-4-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-{1-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-4-phenylbutane-1,4-dione
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-2-oxo-N-(thiophen-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
(3S,4R)-1-[2-chloro-5-(piperidin-1-yl)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
2-methyl-5-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-butyl-4-[2-(ethylamino)pyrimidine-5-carbonyl]-1-methylpiperazin-2-one
7-(cyclopropylmethyl)-N-methyl-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(cyclobutylmethyl)-1-ethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclobutanecarboxamide
{3-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-5-yl}methanol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
ethyl 1-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetyl}piperidine-3-carboxylate
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]pyrrolidine
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide