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methyl 5-methyl-4-{[4-methyl-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl]methyl}-1,2-oxazole-3-carboxylate
(4aR,8aR)-2-(pyrrolidine-1-carbonyl)-7-(thiophene-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
(3S,4R)-1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-propyl-5-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
2-(2-fluorophenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(pyridine-4-carbonyl)-N-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
1-ethyl-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-(2-methylpropyl)-1H-pyrazole
N-(2H-1,3-benzodioxol-5-yl)-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-8-methylquinazolin-4-amine
(4aS,7aR)-1-(3,3-dimethylbutanoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
2-methyl-N-[2-(1-methylpiperidin-4-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(3-methoxy-4-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[3-(2-methyl-1H-imidazol-1-yl)butanoyl]-1-(4-methylphenyl)piperazin-2-one
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]piperidine-3-carboxamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
3-(2H-1,3-benzodioxol-5-yl)-1-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)urea
(1S,6R)-9-[2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-(2,3-dihydro-1-benzofuran-5-ylformamido)-N-(2-methoxyphenyl)propanamide
9-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3,9-diazaspiro[5.6]dodecane
(1S,6R)-9-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-phenylpyrimidin-4-ol
3-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
[(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]urea
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-(1-hydroxypropan-2-yl)-1,2-oxazole-3-carboxamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-(3-methylphenyl)piperidine
5-[1-(2-methoxy-2-methylpropyl)-1H-imidazol-2-yl]-2-(pyridin-2-yl)pyrimidine
5-acetyl-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5,5-dimethyl-3-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,3-oxazolidine-2,4-dione
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(methylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-methoxyethyl)-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
1-(4-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
5-[2-(4-methylpentyl)morpholine-4-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
3-benzyl-4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-(4-methylphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
3-[({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}oxy)methyl]pyridine
4-chloro-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-[4-(2-fluoro-6-methoxyphenyl)phenyl]piperidin-4-ol
2-(3-chlorophenyl)-5-methyl-4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,3-oxazole
N-{[7-(4-cyclopropanecarbonylphenyl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
1-(3-chloro-4-fluorobenzoyl)-3-(2-methoxyphenoxy)azetidine
1-acetyl-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-3-carboxamide
8-fluoro-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)quinoline-2-carboxamide
N-methyl-6-(2,3,4-trimethoxyphenyl)pyridine-2-carboxamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
1-(butane-1-sulfonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-{4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione