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5-(1-cyclopentanecarbonylpiperidin-4-yl)-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-methyl-9-[(1-methyl-1H-imidazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(2-methoxy-5-phenylphenyl)propanamide
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-1H-1,3-benzodiazole
N-[3-(1H-pyrazol-1-yl)phenyl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-[3-(dimethylamino)propyl]-5-[1-(2-methylbutanoyl)piperidin-4-yl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
4-(3-methoxypropyl)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
2-{4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrazine
3-{[(3S)-3-aminopyrrolidin-1-yl]sulfonyl}-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}benzamide
1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(2-methoxypyridine-3-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl]benzamide
6-methyl-2-oxo-N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}-1,2-dihydropyridine-4-carboxamide
3-(benzyloxy)-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
(3aS,6aS)-2-ethyl-1-oxo-5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({8-[(4-hydroxy-3-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-{[3-(hydroxymethyl)-3-(2-methylpropyl)piperidin-1-yl]methyl}-6-methoxyphenol
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
7-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
2-chloro-4,5-difluoro-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
7-(5-chloropyridine-2-carbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[2-chloro-4-(2-methylpyrrolidine-1-carbonyl)phenoxy]-1-methanesulfonylpiperidine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-methoxy-1-(pyridin-2-yl)ethyl]acetamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)cyclobutanamine
1-benzoyl-4-(5-butylpyridine-2-carbonyl)piperazine
2-amino-3-ethyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]methyl}amine
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2,4-dioxoimidazolidin-1-yl)acetamide
2-(1H-1,3-benzodiazol-1-yl)-N-(2-methoxyethyl)propanamide
(3R,4R)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-phenylethyl)carbamoyl]piperidine-4-carboxylate
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]thieno[3,2-d]pyrimidin-4-amine
3-{5-[2-(2,3-dihydro-1H-inden-5-yloxy)propan-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
4-({3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1-ethylpiperidine
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
5-(5-methoxypyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
4-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)quinazoline
6-methyl-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
4-chloro-N-[(4-cyanophenyl)methyl]-1-methyl-1H-pyrazole-3-carboxamide
(4aS,8aR)-1-(3-methylbutyl)-6-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(1H-1,3-benzodiazol-1-yl)-1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]ethan-1-one