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methyl 4-{5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-1,2,4-oxadiazol-3-yl}benzoate
(2S,4S)-4-amino-1-[(4-methylphenyl)methanesulfonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperazin-1-yl}pyrazine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(phenylamino)pyrimidine-5-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-{1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
N-[3-(quinolin-3-yl)propyl]methanesulfonamide
2-(prop-2-en-1-yl)-9-[3-(pyridin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2E)-3-(3,4-dimethoxyphenyl)-1-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)prop-2-en-1-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,6-dihydroxybenzamide
5-fluoro-2-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-N,N-dimethylpyrimidin-4-amine
methyl 2-{4-[(1R,4S)-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-amido]piperidin-1-yl}acetate
2-(2,5-dimethoxyphenyl)-N-[2-(dimethylamino)ethyl]-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}acetamide
4-({5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
dimethyl[(4-methyl-5-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
1-cyclohexyl-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
4-(2-benzyl-3-oxopiperazine-1-carbonyl)-1,2-dihydroquinolin-2-one
3-{4-[(2,4-dimethoxyphenyl)methyl]piperazin-1-yl}-6-methylpyridazine
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]cyclohexanamine
1-benzyl-N-methyl-5-(pyridine-2-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-7-fluoro-3-methyl-1H-indole
N-benzyl-5-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
3-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(2-aminoethyl)-N-[cyclopropyl(pyridin-2-yl)methyl]-N-methylquinazolin-4-amine
2-[6-(2-fluoro-5-methoxyphenyl)pyridin-3-yl]acetic acid
(2S,4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-acetamido-N-ethylpyrrolidine-2-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-4-carboxylate
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})amine
5-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
4-{4-[(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenyl}-2-methylbut-3-yn-2-ol
3-({2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}benzamide
(1S,5R)-3-[2-(5-acetylthiophen-3-yl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 6-(2-cyclopentylacetyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(2-aminoacetyl)-5-benzyl-1-(3-methoxyphenyl)piperazin-2-one
4-(1-ethyl-1H-pyrazole-5-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-(oxolan-3-yl)piperidin-4-amine
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]methanesulfonamide
2-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}propan-1-ol
1-[(3-fluorophenyl)methyl]-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
2-(2,4-dichlorophenoxy)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2,6-difluoro-3-methoxy-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidin-4-amine
2-cyclopentyl-8-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2-methylphenyl)-3-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-1,2,4-triazine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-ol
1-methyl-N-[2-(pyridin-3-yl)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(1-benzyl-1H-imidazol-2-yl)-1-(4-methylbenzoyl)piperidine