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1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(4S)-1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3,3,4-trimethylpiperidin-4-ol
1-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2,6-dimethylpyrimidine-4-carbonyl)pyrrolidin-3-yl]methanol
3-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
(4aS,8aR)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
3-[4-phenyl-1-(1H-1,2,4-triazol-5-ylmethyl)-1H-imidazol-5-yl]quinoline
2-amino-N,6-dimethyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]pyrimidine-4-carboxamide
1-(2-cyclohexylethyl)-N-methyl-N-(oxolan-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-(2-cyclopropylacetyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
3,5-dimethyl-4-[5-(thiophene-3-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
5-ethyl-N-[2-(1H-indol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1,4-oxazepan-6-ol
N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2,3-dihydro-1-benzofuran-5-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[2-(methylsulfanyl)acetyl]-decahydro-1,6-naphthyridin-2-one
ethyl 4-[6-(3-chloro-2-fluorobenzoyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
(3S)-3-methyl-1-(2-methylpropyl)-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
6-[5-(morpholine-4-carbonyl)pyridin-2-yl]quinoline
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclopentyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-tert-butyl-7,7-dimethyl-N-[(trimethylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydroquinazolin-5-amine
N-(cyclopropylmethyl)-4-{methyl[2-(1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide
N,N-dimethyl-2-{[(2-methyl-1-benzofuran-7-yl)formamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-{4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carbonitrile
[(1,2-dimethyl-1H-imidazol-5-yl)methyl]({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl})amine
2-[1-cyclopentyl-4-(naphthalen-1-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(4-methyl-1H-imidazole-2-carbonyl)-1,4-diazepan-6-ol
4-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
(3aR,6aR)-2-cyclopentyl-5-[(4-methyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[2-(3-methoxyphenyl)azetidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-{[4-(6-methoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
3-(2-methoxyethyl)-1-[3-(pyridin-2-yl)propanoyl]piperidine-3-carboxylic acid
3-methyl-7-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-{5-[3-(3-methylphenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
(3R,4R)-4-(azepan-1-yl)-1-(2,2-diphenylethyl)piperidin-3-ol
1-[(2-chloro-4-fluorophenyl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
1-[(1-benzylpyrrolidin-3-yl)methyl]-3-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(2-chlorophenyl)piperazin-2-one
2-(2-aminopyrimidin-5-yl)-N-[2-methyl-1-(pyridin-3-yl)propyl]quinoline-4-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-(4-{[(4-phenyloxan-4-yl)methyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-(piperidin-1-yl)benzoyl]pyrrolidin-3-yl]methanol
5-(butylamino)-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2E)-3-(4-methoxyphenyl)-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-6-methylphenol
(2S,4R)-1-[(2-hydroxy-3-methoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
2-(3,5-dimethyl-4-{[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
5-benzyl-4-cyclopropanecarbonyl-1-(4-methylphenyl)piperazin-2-one