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{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
[(5-ethylpyridin-2-yl)methyl](furan-2-ylmethyl)(3-methylbutan-2-yl)amine
N-(pyridin-2-ylmethyl)-1-(quinoline-3-carbonyl)piperazine-2-carboxamide
3-fluoro-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
methyl (2R,4S)-1-(5-chloro-2-methoxybenzenesulfonyl)-4-hydroxypiperidine-2-carboxylate
6-[4-(3,5-dimethyl-1H-indole-2-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(3S,4R)-1-[2-(4-phenylphenyl)acetyl]-4-propylpyrrolidin-3-yl]acetamide
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2,6-dimethoxy-4-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
4-(2-aminopyridine-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(4-ethoxyphenyl)propyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-[2-(3-methoxyphenyl)phenyl]-1-propylpiperidine-4-carboxamide
2-(3,5-dimethyl-4-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
3-(2-ethylbutyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-{[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(4-methylpentyl)morpholine
1-(3-methylbenzoyl)-3-(naphthalene-1-carbonyl)piperidine
5-(cyclopropylmethyl)-1-(3-fluorophenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}pyridine
3,3-diethyl-1-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)urea
2-amino-4-(3,4-dihydroxyphenyl)-6-(4-fluorophenyl)pyridine-3-carbonitrile
1-(2-methoxyethyl)-8-(propan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-benzyl-4-(2-ethoxypyridine-3-carbonyl)-1,4-diazepan-6-ol
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one
4-(4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-2-oxopiperazin-1-yl)benzonitrile
3-[(3R,4S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methylazepane
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
2-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
3-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
methyl 4-(4-methanesulfonylphenyl)-1H-pyrrole-2-carboxylate
(3R,4R)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3,4-dimethylpyrrolidin-3-ol
1-(4-methoxybenzoyl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazine
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(1-methoxybutan-2-yl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
3-(4-benzyl-1H-pyrazol-5-yl)-1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidine
2,6-difluoro-4-methoxy-N-(1,2-oxazol-3-ylmethyl)benzamide
N,N-dimethyl-4-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(quinolin-7-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(6-chloropyridazin-3-yl)-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
3-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
(1R,3S,5S)-8-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
5-{2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(cyclopentylmethyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine