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(1S,5R)-6-methanesulfonyl-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1'-(1-ethyl-1H-pyrazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 1-(2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}acetyl)piperidine-2-carboxylate
ethyl 1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
2-[2-(3,5-dimethylbenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
2-[1-(2,2-dimethylpent-4-en-1-yl)piperidin-4-yl]-N-methylacetamide
methyl 3-(cyclobutylmethoxy)-5-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]benzoate
1-[2-(tert-butylsulfanyl)ethyl]-4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazole
1-ethyl-N-methyl-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(1,3-dimethylpyrrolidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-benzyl-1-[1-(furan-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
N-benzyl({6-[(propan-2-yl)amino]pyridin-3-yl}amino)sulfonamide
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrazine-2-carboxamide
2-[3-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-(4-methyl-1-propyl-1H-pyrazol-5-yl)acetamide
1-(azepan-1-yl)-3-[2-(4-chlorophenyl)-1H-imidazol-1-yl]propan-2-ol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}oxane-2-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-{2-cyclobutyl-1-methyl-7-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
3-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-3-yl]propanamide
(3S,4R)-1-[2-(dimethylamino)benzoyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
(4aS,7aR)-1-[(5-phenylthiophen-2-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
methyl 3-(2-methoxybenzamido)-5-{[(1-methyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
N-benzyl-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(2S,4R)-4-amino-N-ethyl-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
5-methyl-2-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}phenol
methyl(3-phenylpropyl){[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}amine
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-6-methoxyphenol
N-(6-phenoxypyridin-3-yl)-1-(1,3-thiazol-5-ylmethyl)piperidine-2-carboxamide
(2S,4R)-N-methyl-1-(propan-2-yl)-4-({[4-(propan-2-yl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-4-(piperidin-3-yl)benzamide
5-acetyl-N-[(3-chlorophenyl)methyl]-6-methyl-2-oxo-N-propyl-1,2-dihydropyridine-3-carboxamide
N-butyl-N-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
2-{1-benzyl-4-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-1-yl]acetamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}propan-1-one
1-(2-amino-9H-purin-6-yl)-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepan-6-ol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(4-methoxy-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-amine
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-1H-indazole-3-carboxamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
(3S,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carbonitrile