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8-[(3-chloro-4-methoxyphenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aS,8aR)-6-[3-(1-methyl-1H-pyrrol-2-yl)propanoyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
4-benzyl-3-ethyl-1-(1H-imidazole-2-carbonyl)-1,4-diazepan-5-one
N-ethyl-1-{2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidine-3-carboxamide
2,5-dimethyl-3-[4-(thiophen-3-ylmethyl)piperazin-1-yl]pyrazine
1-[2-(4-methoxyphenyl)ethyl]-8-(1-methoxypropan-2-yl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-9H-fluorene-9-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
(3aS,6aR)-N-(4-methylphenyl)-2-oxo-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
2-amino-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one
N-(6-cyanopyridin-3-yl)-4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)benzamide
N-(furan-2-ylmethyl)-2-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]acetamide
7-(5-chloropyridin-2-yl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(2-methylpropanesulfonyl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
1-{4-[4-chloro-2-(3-propoxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
ethyl 4-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-amido]piperidine-1-carboxylate
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-[2-(3,4-dimethoxyphenyl)-4-methylphenoxy]acetamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]acetamide
4-(7-chloro-4-methylquinolin-2-yl)-1-ethyl-3-methylpiperazin-2-one
2-(adamantan-1-yl)-5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrimidin-4-ol
4,4-difluoro-N-(6-methoxyquinolin-8-yl)piperidine-1-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(4aS,8aR)-6-(3-chloro-5-fluorobenzoyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N,N-diethyl-1-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propane-1,2-dione
4-(1-acetylpiperidin-4-yl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-methoxy-3-(3,4,5-trimethoxyphenyl)quinoline
3-[({1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
N-[1-({[(2,4-dimethoxyphenyl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
1-(4-fluorophenyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]cyclopropane-1-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)acetamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-(4-methyl-1,4-diazepan-1-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-(4-methyl-1H-pyrazol-1-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
(3R,5S)-N3-(4-fluorophenyl)-N5-(3-methoxypropyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
1-[(4-chlorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
benzyl({[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
1-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-(naphthalen-2-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-(methoxymethyl)-N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}furan-2-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-methylfuran-2-carboxamide
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-(3-fluoro-4-methoxyphenyl)acetic acid
6-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one