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6-methyl-2-[({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)methyl]quinolin-4-ol
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
5-methyl-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-(2-methylpropyl)-5-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
1-benzyl-N-(butan-2-yl)-5-methyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}morpholin-2-yl)ethan-1-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{[2-(2-methylpropanesulfonyl)ethyl]amino}pyrimidine-5-carboxylic acid
2-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N,2,4-trimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-(methylamino)pyrimidine-5-carboxamide
1-(3,4-difluorophenyl)-5-[(4-methanesulfonylphenyl)methyl]-1H-1,2,4-triazole
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]piperidine-3-carboxamide
N-[(3S)-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl]acetamide
N,N-dimethyl-2-{[4-(pyrrolidin-1-yl)butanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
5-[(2E)-but-2-en-1-yl]-3-(oxan-4-yl)-1H-1,2,4-triazole
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(2-hydroxyethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}sulfonyl)azepane
N-methyl-2-{3-oxo-1-[2-(quinazolin-4-yloxy)acetyl]piperazin-2-yl}acetamide
[1-(2,6-dimethylphenoxy)propan-2-yl]({[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl})amine
N-[(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-4-carboxamide
N-cyclopropyl-4-methyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)benzamide
N-({7-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-2-(thiophen-3-yl)acetamide
4-(1,5-dimethyl-1H-indole-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
methyl 3-[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]propanoate
N-(propan-2-yl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-ethylpyridin-2-yl)methyl]piperidine-3-carboxamide
1-[(2S)-2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-1-yl]ethan-1-one
(2S,4R)-4-amino-N-ethyl-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
2-hydroxy-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
5-[4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylacetamide
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-1-[(4-methoxyphenyl)methyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N3-[(3-chlorophenyl)methyl]-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5,6-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2-(2-oxoazepan-1-yl)acetamide
1-(2-methoxyethyl)-4-oxo-N3-(2-phenylethyl)-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(cyclopropylmethyl)-8-(4-phenoxybutanoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-methoxyphenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclopentyl-4-(5-methanesulfonyl-2-methylpyrimidin-4-yl)piperazin-2-one
4-{[2-(4-methylpyrimidin-2-yl)phenyl]methyl}morpholine
2-amino-N,3-diethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide