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5-benzyl-4-(1H-imidazole-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
(3R,5S)-5-(morpholine-4-carbonyl)-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
methyl 1-{9-methoxy-7-oxo-3-[(2,4,5-trimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
4-chloro-5-{[ethyl(oxan-4-yl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2-methoxyacetamide
1-[2-(dimethylamino)ethyl]-N-methyl-6-oxo-N-[3-(pyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-cyclohexyl-4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}piperidine-1-carboxamide
ethyl 4-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)piperidine-1-carboxylate
N-(furan-2-ylmethyl)-N-methyl-3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzamide
1-(cyclopent-3-en-1-yl)-5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
2-amino-6-tert-butyl-4-(1H-imidazol-4-yl)pyridine-3-carbonitrile
ethyl 1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(9H-purin-2-yl)piperidine-4-carboxylic acid
N-({3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]phenyl}methyl)acetamide
1-(2,6-dimethylpyridin-4-yl)-4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
2-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-methyl-2-[1-(3-methylfuran-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]pyridine
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
N-ethyl-N-(4-hydroxybutyl)-3-(1H-pyrazol-4-yl)benzamide
1-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-(1-methyl-1H-indol-3-yl)ethan-1-one
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-oxopropyl)urea
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(morpholine-4-carbonyl)piperazin-1-yl]ethan-1-one
4-(1-methanesulfonylpiperidin-3-yl)benzoic acid
(2R,3R,6R)-3-(4-methylphenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(1H-pyrazol-3-yl)piperidine
ethyl 1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-(oxan-3-ylmethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
(3S,4S)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(1H-imidazol-2-yl)pyrrolidine-3-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(quinolin-5-ylmethyl)piperidin-3-yl]propanamide
(2S)-4-methyl-2-(propan-2-yl)-1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
1,6-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[7-(cyclohex-3-en-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
6-(furan-3-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
ethyl 1-{1-cyclopentyl-5-[(2-methylpropyl)carbamoyl]-4-oxo-1,4-dihydropyridine-3-carbonyl}piperidine-3-carboxylate
8-(2-methyl-1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-(propan-2-yl)piperidin-4-amine
1-[(3-fluorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-{1-[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl]piperidin-3-yl}-1,3-benzoxazole
3-(2H-1,3-benzodioxol-5-yl)-N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]propanamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-6-(2-methoxyethyl)-3-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)-N-[3-(morpholin-4-yl)propyl]pyridine-3-carboxamide
3-[1-(furan-3-ylmethyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1H-indazole
N,N-bis(2-hydroxyethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)pyrazine
2-{[4-(5-chloro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine