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(3S,4S)-4-(morpholin-4-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-ol
2-[1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)azetidin-3-yl]pyridine
7-(1-ethyl-1H-pyrazole-3-carbonyl)-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{2-[1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-(dicyclopropylmethyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-acetyl-N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]piperidine-4-carboxamide
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[(3R,4S)-3-acetamido-4-propylpyrrolidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
1-[(2,5-dimethoxyphenyl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
1-cyclohexyl-3-(cyclopropylmethyl)-N-(1,3-dihydroxypropan-2-yl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(cyclohexylmethyl)-2-(methoxymethyl)-N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
1-{4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-(4-{4-methoxy-2-[2-(pyridin-3-yl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
1-{2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-methyl-1,3,4-oxadiazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(3aS,6aS)-2-methyl-5-(pyrrolidine-1-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
9-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-fluoro-N-methyl-4-(morpholin-4-yl)pyrimidin-2-amine
(2S,4S)-4-amino-1-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(2-methoxyethyl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
3-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-2-yl}propanoic acid
(2R)-2-acetamido-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}propanamide
3-{[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamido]methyl}-1,2,4-oxadiazole-5-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
2-(5-methylpyrazine-2-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-1-one
2-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
[3-benzyl-1-(3-chloropyridin-2-yl)piperidin-3-yl]methanol
[3-benzyl-1-(2-methoxy-5-methylbenzenesulfonyl)piperidin-3-yl]methanol
3-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(dimethylamino)ethan-1-one
3-(2-amino-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-[2-(phenylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(pyrimidin-4-yl)ethyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(3S,4S)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-({[2-(dimethylamino)ethyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)amino}methyl)-6-methoxyphenol
(3R)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3,4,4-trimethylpyrrolidin-3-ol
2-methyl-4-{4-[4-(1H-1,2,3,4-tetrazol-5-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-[5-cyclopropyl-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]-4-[2-(trifluoromethyl)phenyl]pyrimidine
N,N-dimethyl-2-[(1S,5R)-6-phenylmethanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-{1-[4-(dimethylamino)butanoyl]piperidin-3-yl}benzoic acid
6,7-dimethoxy-2-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(4aR,7aS)-1-(2-hydroxyethyl)-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-ethanesulfonamidobenzamide