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4-(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
N,N-dimethyl-2-(2-oxo-5,5-diphenylpiperidin-1-yl)ethane-1-sulfonamide
1-[2-(azepan-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
[(3S,4S)-1-{[4-(4-chlorophenyl)phenyl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methanol
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
5-(5-chloro-7-methoxy-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(oxan-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-hydroxyethyl)-9-[(5-methylnaphthalen-1-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-5-(2,6-dimethylphenoxymethyl)-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
1-[2-(cyclopropylcarbamoyl)ethyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-benzyl-1-ethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
9-cyclobutanecarbonyl-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
7-(cyclopropylmethyl)-2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
5-(1-ethyl-1H-pyrazol-4-yl)-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(2Z)-2-fluoro-1-{3-[5-(4-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
N-(2-methoxyethyl)-3-(piperidin-1-yl)-N-(thiophen-2-ylmethyl)propanamide
5-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecane
3-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-cyclohexylpropanamide
2-{1-benzyl-4-[(4-chlorophenyl)methyl]piperazin-2-yl}ethan-1-ol
4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-3-ethylpiperazin-2-one
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-2-amine
4-cyano-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-pyrrole-2-carboxamide
3-{5-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(3S,4R)-4-(2-methylphenyl)-1-(quinoxaline-5-carbonyl)pyrrolidine-3-carboxylic acid
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-methyl-1-[4-(methylsulfanyl)phenyl]urea
3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(2-methylphenyl)-3-[1-(1-propanoylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}-N-benzyl-N-methylpropanamide
N-methyl-N-[2-methyl-3-(pyrrolidin-1-yl)propyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-N-(propan-2-yl)benzamide
(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-3-yl)methanamine
[(1-cyclopentylpiperidin-4-yl)methyl][(2,6-dimethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
{3-[(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
6-(1-benzothiophen-3-yl)-2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]pyridine-3-carboxamide
1-(2-methoxyethyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidine-4-carboxamide
1-cyclohexyl-4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-methyl-2-[4-(morpholin-4-yl)-2-{[2-(morpholin-4-yl)ethyl]amino}pyrimidin-5-yl]propanoic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]thiophene-3-sulfonamide
4-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]thiomorpholine
N-(3-methoxyphenyl)-3-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}propanamide