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3-{2-[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}-1-methylpyrrolidin-2-one
N-butyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(4-methylphenyl)methyl]acetamide
2-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
N-benzyl-3-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-methylpropanamide
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-[4-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-5-{2-[2-({7-methylthieno[3,2-d]pyrimidin-4-yl}amino)ethyl]morpholin-4-yl}-2,3-dihydropyridazin-3-one
(3R,4R)-4-amino-1-{[4-(3,4-dimethylphenoxy)phenyl]methyl}piperidin-3-ol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)piperidin-2-one
4-[2-amino-3-cyano-6-(6-methoxypyridin-3-yl)pyridin-4-yl]benzoic acid
(3S,4S)-1-(cyclopropanesulfonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-({1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
2-(adamantan-1-yl)-N-ethyl-N-(oxan-4-yl)acetamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
5-methoxy-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-1H-indole-2-carboxamide
2-[5-(methoxymethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
9-[2-(1H-indol-3-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
ethyl 1-[2-(2-methoxyphenoxy)acetyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
1-[4-(propan-2-yl)piperazin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-(1-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
1-(thiomorpholin-4-yl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-(2-cyclopentyl-2-phenylethyl)pyridine-3-carboxamide
(2S,4S)-N-ethyl-4-(furan-3-amido)-1-[3-(1H-pyrrol-1-yl)propanoyl]pyrrolidine-2-carboxamide
1-(4-chloro-2-fluorophenyl)-3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
9-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperazine-1-carboxylate
1-[(2-chloro-4-fluorophenyl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
5-(4-fluoro-2-methoxyphenyl)-1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazole
2-(furan-2-yl)-5-{[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrimidine
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(4-fluorophenyl)ethan-1-one
2-(2-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
9-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-chloro-N-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzamide
methyl 1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
1-(cyclohexylmethyl)-N-(3-hydroxy-2,2-dimethylpropyl)-6-oxopiperidine-3-carboxamide
N,N-dimethyl-2-{[3-(N-methylmethanesulfonamido)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
3-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-indol-2-one
3-{[1-(3-chloro-4-methylphenyl)piperidin-4-yl](methyl)amino}propanamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
3-(4-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2,5-dimethoxyphenyl)acetamide
N,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-propyl-1-benzofuran-2-carboxamide
2-chloro-N-(2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}ethyl)benzamide
5-{2-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}quinoline
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-(1,3-benzothiazol-2-yl)-N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine