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(2S)-1-({3-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-2-(propan-2-yl)piperazine
3-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-{3-methyl-4-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazol-1-yl}ethan-1-ol
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(hydroxymethyl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
N-(2-methoxy-5-methylphenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
9-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-methyl-4-[5-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)thiophen-2-yl]but-3-yn-2-ol
1-(3-methoxypropyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
1-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-ethyl-3-{[(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)carbamoyl]amino}-2-methylbenzamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
7-[(4-fluorophenyl)methyl]-2-(4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
4-(6-aminopyridine-3-carbonyl)-1-(4-chlorophenyl)-5-methylpiperazin-2-one
methyl (2S)-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
N-(4-methoxyphenyl)-1-[(2-methoxyphenyl)methyl]piperidin-3-amine
2-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
4-(5-fluoro-2-methoxyphenyl)-6-(1H-pyrazol-1-yl)pyrimidine
N-({7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-(3,4-difluorophenyl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
5-(4-chlorophenyl)-3-(morpholin-4-yl)-1,2,4-triazine
1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}ethan-1-one
2-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2,4-dimethoxy-3-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{4-[(2,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
2-ethoxy-4-[(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
5-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]-2,3-dimethylbenzene-1-sulfonamide
N3-[(2-benzyl-1,3-thiazol-4-yl)methyl]-N5-cyclohexyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-methoxybenzoyl)piperazine
1-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
[7-(7-chloroquinolin-4-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(2H-1,3-benzodioxol-5-yl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
6-[4-(2-aminopyrimidin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-[2-(azepan-1-yl)ethyl]-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(1H-pyrazol-5-ylmethyl)amino]pyridine-3-carboxamide
4-[2-(3-{3-[2-(methylsulfanyl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)ethyl]morpholine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-indazole-3-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-4-(piperidin-3-yl)benzamide
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide