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1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-(2,5-difluorobenzoyl)-1-(3,5-dimethylfuran-2-carbonyl)piperidine
N-methyl-N-(1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-2-phenylethyl)thiophene-3-carboxamide
4-(1-{6-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine-3-carbonyl}piperidin-4-yl)morpholine
3-{1-[2-(3-methoxyphenyl)phenyl]-1H-imidazol-2-yl}pyridine
2-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-N-methylacetamide
8-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione
(3aR,5S,6S,7aS)-2-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-octahydro-1H-isoindole-5,6-diol
3-[(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
4-({2-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(1H-imidazol-4-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
8-chloro-2-(furan-2-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)quinoline-4-carboxamide
5-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}pyrazin-2-ol
1-[1-(5-chloro-2-fluorobenzoyl)-4-phenylpiperidin-4-yl]ethan-1-one
6-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl[(4-{2-[1-(4-methylbenzoyl)piperidin-2-yl]ethoxy}phenyl)methyl](quinolin-5-ylmethyl)amine
N,N,7,8-tetramethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(oxolan-3-yl)ethyl]-1,3-oxazole-4-carboxamide
2-{4-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenoxy}ethan-1-ol
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
(4S)-1-(1H-imidazol-4-ylmethyl)-3,3,4-trimethylpiperidin-4-ol
1-(1,3-benzothiazol-2-yl)-N-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-amine
1-(3-{[3-(pyrrolidine-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
7-[(3-phenoxyphenyl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
4-(1,3-benzothiazol-2-yl)-1-methylpiperazine-2-carboxylic acid
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}butanamide
[1-(cyclohex-1-ene-1-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
4-({3-[(3-chlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}methyl)-1λ6-thiane-1,1-dione
1-(4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-oxobutyl)piperidin-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]urea
3-hexyl-8-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(isoquinolin-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
9-[(2S)-2-amino-2-cyclopropylacetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]butanamide
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(methylsulfanyl)propanamide
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-[(4-fluorophenyl)formamido]-N-methylpropanamide
3-(3-hydroxyquinoxalin-2-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
2-(methoxymethyl)-5-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}pyrimidine
2-chloro-5-[2-fluoro-6-(propan-2-yloxy)phenyl]pyrazine
2-[4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]acetamide
N4-{3-[ethyl(methyl)amino]-2-methylpropyl}-5,6-dimethylpyrimidine-2,4-diamine
5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
(3aS,6aS)-2-methyl-5-{2-[3-(trifluoromethyl)phenyl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
(3S,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-benzyl-2-(3-fluorophenyl)-3-oxopiperazine-1-sulfonamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1H-indole-5-carboxamide