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1-[(3-methylthiophen-2-yl)methyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-(4-methoxyphenyl)-5-{[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidine
N-(2H-1,3-benzodioxol-5-yl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carboxamide
4-(1H-pyrazol-4-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]butan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
5-(3-methylbutyl)-5-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(methylsulfanyl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-4-amine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amine
6-(5-chloro-3-methyl-1H-indole-2-carbonyl)-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-chloro-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)benzamide
2-methyl-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}-1,3-thiazole-4-carboxamide
N-cyclopentyl-3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanamide
1-methyl-4-{1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
N-[(6-methylpyridin-2-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)adamantane-1-carboxamide
6-{[(cyclopropylmethyl)(propyl)amino]methyl}-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
4-[(2,4-dimethoxyphenyl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 4-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
3-{[(1-methanesulfonylpiperidin-3-yl)methyl]amino}-N-(pyridin-3-yl)propanamide
2-cyclopentyl-1-[4-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(3-fluoro-4-methoxybenzoyl)piperidine
N-(1-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
5-{2-[(2,3-dihydro-1H-inden-2-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine
[1-(6-methoxypyrimidin-4-yl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
2-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-5-methoxy-1,4-dihydropyridin-4-one
5-(morpholin-4-ylmethyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)furan-3-carboxamide
2,3,5-trimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-oxo-1-{3-[(pyridin-3-yl)amino]propyl}pyrrolidine-3-carboxylic acid
1-[(2-methoxyphenyl)methyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-(thiophen-2-ylmethyl)pyrimidine-5-carboxamide
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1H-pyrazole-3-carboxylic acid
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(2-hydroxyethoxy)ethyl]acetamide
1-(3-hydroxypropyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
N-{2-[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
4-({3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzoic acid
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N,2-diethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]pyrimidine-5-carboxamide
1-[(3aR,6aR)-3a-(2,5-dihydro-1H-pyrrole-1-carbonyl)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methoxyethan-1-one
N-[2-(5-methyl-4-{[3-(4-methyl-1,3-thiazol-5-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]benzamide
3-methyl-N-(1,2-oxazol-3-ylmethyl)-5-propyl-1-benzofuran-2-carboxamide
4-(2-methoxy-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)-1-(propan-2-yl)piperidine
2-(2-methoxyethyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N-{[1-(dimethylamino)cyclohexyl]methyl}-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
methyl N-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}carbamate