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N-cyclobutyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3S,4R)-1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
(3S,4S)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
{[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)(propan-2-yl)amine
7-(2-propoxybenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-4-sulfamoylbenzamide
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
1-sulfamoyl-4-[2-(thiophen-2-yl)acetyl]-1,4-diazepane-6-carboxylic acid
7-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
(4aS,7aR)-6,6-dioxo-N-propyl-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2R,3R,6R)-5-(1H-imidazol-4-ylmethyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)-1,3-thiazole
N-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-2-methylpropanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(1H-pyrazol-3-yl)benzamide
N-cyclopentyl-N-{[3-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
N-(pyridin-3-ylmethyl)-N-[(2,3,4-trifluorophenyl)methyl]cyclopropanamine
3-(1H-1,2,3-benzotriazol-5-yl)-1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}urea
4-benzyl-3-ethyl-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-5-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(quinolin-5-ylmethyl)acetamide
1-{4-[2-(3-phenylpropyl)morpholin-4-yl]piperidin-1-yl}ethan-1-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(thiophene-2-carbonyl)-1,4-diazepan-5-one
1'-(1-ethyl-1H-pyrazole-5-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(1,3-benzothiazol-2-yl)-4-(3,5-dimethoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methoxy-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-2-(2,4-difluorophenyl)acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-[4-(trifluoromethyl)benzoyl]piperidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}piperidin-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,5-dimethyl-1-phenyl-1H-pyrrole-3-carboxamide
2-(2-chlorophenyl)-N-(2-fluoroethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3R,4R)-1-{2-[(dimethylamino)methyl]benzoyl}-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
methyl 6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-(methylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3ar,6ar)-N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-1,2-dihydroquinolin-2-one
2-[2-(1H-imidazol-1-yl)ethyl]-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
5-[(4-benzylpiperidin-1-yl)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
4-[(2H-1,3-benzodioxol-4-ylmethyl)amino]-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-2-one
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}phenyl)-1,4-diazepane-1-carboxamide
4-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-amine
1-{3-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]phenyl}propan-1-one
2-ethyl-N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-ethyl-2-(1H-indol-3-yl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-methoxy-4-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)phenol
(3S)-N,N-dimethyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
2-({[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
3-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide